Structure information

δ receptor

PROTEIN CLASS

Class A (Rhodopsin)

PDB CODE

8Y45

SPECIES

Homo sapiens

RESOLUTION

3.450

PREFERRED CHAIN

A

REFERENCE

PUBLICATION DATE

Nov. 27, 2024

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Ligand Interaction Browser

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Ligand Amino Acid Generic Number Segment Interaction Type
Ligand Amino Acid Generic Number Segment Interaction Type
ADL5859 Y129 3.33x33 TM3 polar (hydrogen bond)
ADL5859 M132 3.36x36 TM3 polar (hydrogen bond)
ADL5859 K214 5.39x40 TM5 Van der Waals
ADL5859 I277 6.51x51 TM6 hydrophobic
ADL5859 I277 6.51x51 TM6 Van der Waals
ADL5859 V281 6.55x55 TM6 hydrophobic
ADL5859 V281 6.55x55 TM6 Van der Waals
ADL5859 W284 6.58x58 TM6 Van der Waals
ADL5859 W284 6.58x58 TM6 hydrophobic
ADL5859 L300 7.35x34 TM7 hydrophobic
ADL5859 L300 7.35x34 TM7 Van der Waals
ADL5859 I304 7.39x38 TM7 hydrophobic
ADL5859 I304 7.39x38 TM7 Van der Waals
ADL5859 Y308 7.43x42 TM7 hydrophobic
ADL5859 Y308 7.43x42 TM7 Van der Waals

Ligands

ADL5859

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Residue Diagrams

V N G L L G V A C V A S Y L A T I A I A 1 F N L A L A D A L A T S T L P F Q S A K 2 M T L T F I S T F M N Y Y D I S L V A K 3 A K L I N I C I W V L A S G V G V P I M 4 Y C V T I I L I P V V F A F L F V C I K T 5 L V V V G A F V V C W A P I H I F V I V 6 V P N L S S N A Y G L A I C L H L A A 7
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ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 V T R P R D G A V V C M L Q F P S ECL2ICL3 R L L S G ICL3ECL3 D I D R R ECL3N-term M E P A P S A G A E L Q P P L F A N A S D A Y P S A C P S A G A N A S G P P N-termC-term P C G R P D P S S F S R A R E A T A R E R V T A C T P S D G P G G G A A A C-term G A R S A S S L A L A I A I T A L Y S A V C A V G L L G N V L V M F G I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S A K Y L M E G E L L C K A V L S I D Y Y N M F T S I F T L T M M S V D R Y I A V C H T P A K A K L I N I C I W V L A S G V G V P I M V M A P S W Y W D T V T K I C V F L F A F V V P I L I I T V C Y G L M L L R L R S V S K E K D R S L R R I T R M V L V V V G A F V V C W A P I H I F V I V W T L V D P L V V A A L H L C I A L G Y A N S S L N P V L Y A F L D E N F R Q F K R C L C R K
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Residue Table


GPCRdb(A)
GPCRdb(A)
δ receptor
TM3
3x33 3.33x33 Y129
3x36 3.36x36 M132
TM5
5x40 5.39x40 K214
TM6
6x51 6.51x51 I277
6x55 6.55x55 V281
6x58 6.58x58 W284
TM7
7x34 7.35x34 L300
7x38 7.39x38 I304
7x42 7.43x42 Y308