ArrestinDb

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

Ligands				Receptor	Activity									Chemical information
Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

A(Δ10/15C)INSL3	282	None	0	Human	Binding	pKi	=	-	8.32	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/20570702
A(10-24)INSL3	190	None	0	Human	Binding	pKi	=	-	8.67	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18434306
A(4-24)(B7-24)H2	202	None	0	Human	Binding	pKi	=	-	6.00	-9	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/21878627
A(9-26)INSL3	214	None	0	Human	Binding	pKi	=	-	9.14	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18434306
A(C10/15S)INSL3	233	None	0	Human	Binding	pKi	=	-	8.59	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/20570702
cyclic INSL3 B-chain analogue 6	1279	None	0	Human	Binding	pKi	=	-	6.65	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/17120268
europium-labelled INSL3	1599	None	0	Human	Binding	pKd	=	-	9.00	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18529069
INSL3	2044	None	0	Human	Binding	pKd	=	-	10.35	16982	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18434306
INSL3	2044	None	0	Human	Binding	pKi	=	-	9.52	16982	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/15649866
INSL3	2044	None	0	Human	Binding	pKi	=	-	9.52	16982	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18434306
INSL3 [A(5-26):B(7-27)]	2045	None	0	Human	Binding	pKi	=	-	7.80	-	1	Receptor binding	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/22654853
INSL3 B chain dimer analogue 8	2047	None	0	Human	Binding	pKi	=	-	8.50	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/20560146
INSL3 B-chain analogue	2046	None	0	Human	Binding	pKi	=	-	5.10	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/16547350
NanoLuc-INSL3	2731	None	0	Human	Binding	pKd	=	-	8.70	-	1	Receptor binding affinity	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/24056075
relaxin	3302	None	0	Human	Binding	pKi	None	-	7.80	-39	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/15649866
relaxin	3303	None	0	Human	Binding	pKi	None	-	7.90	-15	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/15649866
relaxin	3305	None	0	Human	Binding	pKi	=	-	8.39	-40	3	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/15649866
relaxin	3305	None	0	Human	Binding	pKi	=	-	8.39	-40	3	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/18434306
relaxin-1	3306	None	0	Human	Binding	pKi	None	-	8.80	-	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/16411781
relaxin-3	3307	None	0	Human	Binding	pKi	None	-	7.00	-81	4	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/16411781

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Ligand source activities (1 row/activity)