Ligand source activities (1 row/activity)



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Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
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name		 GPCRdb
ID		 #Vendors

 Reference
ligand		 Fold
selectivity		 # Tested
GPCRs		 Species

 p-value
(-log)		 Activity
Type		 Activity
Relation		 Activity
Value		 AssayType

 Assay
Description		 Source

 Mol
weight		 Rot
Bonds		 H don

 H acc

 LogP

 Smiles

 DOI
165271 98756 33 None - 1 Human 10.5 pEC50 = 10.5 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 141 3 3 3 -0.7 N[C@H](CO)Cc1c[nH]cn1 nan
CHEMBL278081 98756 33 None - 1 Human 10.5 pEC50 = 10.5 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 141 3 3 3 -0.7 N[C@H](CO)Cc1c[nH]cn1 nan
CHEMBL4517318 213971 68 None - 1 Human 9.8 pEC50 = 9.8 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43CO)[C@@H]1CCC2=O nan
70914 16476 99 None - 1 Human 9.6 pEC50 = 9.6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 189 5 3 3 -0.6 CC(=O)N[C@@H](CCC(=O)O)C(=O)O nan
CHEMBL1234751 16476 99 None - 1 Human 9.6 pEC50 = 9.6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 189 5 3 3 -0.6 CC(=O)N[C@@H](CCC(=O)O)C(=O)O nan
440832 14106 8 None - 1 Human 9.4 pEC50 = 9.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 271 1 4 4 3.2 Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 nan
CHEMBL1197905 14106 8 None - 1 Human 9.4 pEC50 = 9.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 271 1 4 4 3.2 Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 nan
CHEMBL591036 14106 8 None - 1 Human 9.4 pEC50 = 9.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 271 1 4 4 3.2 Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 nan
10204 71467 27 None - 1 Human 9.2 pEC50 = 9.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 1 2 3.9 C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O nan
CHEMBL196228 71467 27 None - 1 Human 9.2 pEC50 = 9.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 1 2 3.9 C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O nan
222865 16397 31 None - 1 Human 9.1 pEC50 = 9.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 0 2 4.2 C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12 nan
CHEMBL1230438 16397 31 None - 1 Human 9.1 pEC50 = 9.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 0 2 4.2 C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12 nan
3812 717 42 None -2 3 Human 8.9 pEC50 = 8.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
439201 717 42 None -2 3 Human 8.9 pEC50 = 8.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
649 717 42 None -2 3 Human 8.9 pEC50 = 8.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
CHEMBL406291 717 42 None -2 3 Human 8.9 pEC50 = 8.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
DB12126 717 42 None -2 3 Human 8.9 pEC50 = 8.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
12025 98594 89 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 85 0 1 1 -0.1 O=C1CCCN1 nan
CHEMBL276849 98594 89 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 85 0 1 1 -0.1 O=C1CCCN1 nan
CHEMBL4556656 214006 44 None - 1 Human 8.7 pEC50 = 8.7 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None O=C(O)[C@@H](O)CO nan
CHEMBL4590792 214019 38 None - 1 Human 6.0 pEC50 = 6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None O=C[C@H](O[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@@H](O)[C@H](O)[C@H](O)CO nan
11163 100702 113 None - 1 Human 5.0 pEC50 = 5.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 132 3 3 3 -1.9 NCC(=O)NCC(=O)O nan
1548897 100702 113 None - 1 Human 5.0 pEC50 = 5.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 132 3 3 3 -1.9 NCC(=O)NCC(=O)O nan
CHEMBL292467 100702 113 None - 1 Human 5.0 pEC50 = 5.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 132 3 3 3 -1.9 NCC(=O)NCC(=O)O nan
171161 67289 49 None - 1 Human 4.9 pEC50 = 4.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 264 7 2 4 1.0 COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1 nan
CHEMBL1882218 67289 49 None - 1 Human 4.9 pEC50 = 4.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 264 7 2 4 1.0 COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1 nan
5460362 101698 66 None - 1 Human 4.9 pEC50 = 4.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 160 3 3 3 -1.1 C[C@@H](N)C(=O)N[C@H](C)C(=O)O nan
6992112 101698 66 None - 1 Human 4.9 pEC50 = 4.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 160 3 3 3 -1.1 C[C@@H](N)C(=O)N[C@H](C)C(=O)O nan
CHEMBL299420 101698 66 None - 1 Human 4.9 pEC50 = 4.9 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 160 3 3 3 -1.1 C[C@@H](N)C(=O)N[C@H](C)C(=O)O nan
1176 208209 97 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 60 0 2 1 -1.0 NC(N)=O nan
CHEMBL985 208209 97 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 60 0 2 1 -1.0 NC(N)=O nan
CHEMBL4574750 214016 18 None - 1 Human 7.6 pEC50 = 7.6 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None Nc1ncnc2c1ncn2C1OC(CO)C2OP(=O)(O)OC21 nan
964 16391 42 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 104 2 2 3 -1.4 O=C(O)C(=O)CO nan
CHEMBL1230192 16391 42 None - 1 Human 6.4 pEC50 = 6.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 104 2 2 3 -1.4 O=C(O)C(=O)CO nan
3636 361 125 None 22908 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 146 4 2 3 -0.5 OC(=O)CCC(=O)C(=O)O nan
51 361 125 None 22908 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 146 4 2 3 -0.5 OC(=O)CCC(=O)C(=O)O nan
CHEMBL1686 361 125 None 22908 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 146 4 2 3 -0.5 OC(=O)CCC(=O)C(=O)O nan
DB08845 361 125 None 22908 2 Human 8.3 pEC50 = 8.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 146 4 2 3 -0.5 OC(=O)CCC(=O)C(=O)O nan
5756 69627 77 None - 1 Human 4.3 pEC50 = 4.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 3 3 2.6 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O nan
CHEMBL193482 69627 77 None - 1 Human 4.3 pEC50 = 4.3 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 288 0 3 3 2.6 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O nan
124072 107535 88 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 372 10 2 6 3.2 COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O nan
CHEMBL318743 107535 88 None - 1 Human 6.2 pEC50 = 6.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 372 10 2 6 3.2 COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O nan
1319 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
4084 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
4635 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
5257127 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
727 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
750 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
CHEMBL773 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
DB00145 1826 130 None 12302 2 Human 7.2 pEC50 = 7.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 75 1 2 2 -1.0 NCC(=O)O nan
CHEMBL4566376 214013 0 None - 1 Human 8.2 pEC50 = 8.2 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL None None None None nan
1055 2994 105 None 2884 2 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 256 14 1 1 5.6 CCCCCCCCCCCCCCCC(=O)O nan
135369651 2994 105 None 2884 2 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 256 14 1 1 5.6 CCCCCCCCCCCCCCCC(=O)O nan
985 2994 105 None 2884 2 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 256 14 1 1 5.6 CCCCCCCCCCCCCCCC(=O)O nan
CHEMBL82293 2994 105 None 2884 2 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 256 14 1 1 5.6 CCCCCCCCCCCCCCCC(=O)O nan
DB03796 2994 105 None 2884 2 Human 8.0 pEC50 = 8.0 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 256 14 1 1 5.6 CCCCCCCCCCCCCCCC(=O)O nan
5282379 194984 69 None 25 4 Human 6.8 pIC50 = 6.8 Functional
Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 300 5 1 1 5.6 CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1 nan
CHEMBL547 194984 69 None 25 4 Human 6.8 pIC50 = 6.8 Functional
Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
ChEMBL 300 5 1 1 5.6 CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1 nan
5756 69627 77 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 288 0 3 3 2.6 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O None
CHEMBL193482 69627 77 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 288 0 3 3 2.6 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O None
10577 217708 0 None - 1 Human 8.4 pEC50 = 8.4 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 488 8 3 7 3.4 C[C@]12CC[C@H]3[C@@H](CCC4=CC(O)=CC=C34)[C@@H]1C[C@@H](OC(=O)CCC(O)=O)[C@@H]2OC(=O)CCC(O)=O None
1319 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
4084 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
4635 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
5257127 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
727 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
750 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
CHEMBL773 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
DB00145 1826 130 None 12302 2 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 75 1 2 2 -1.0 NCC(=O)O None
1176 208209 97 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 60 0 2 1 -1.0 NC(N)=O None
CHEMBL985 208209 97 None - 1 Human 8.1 pEC50 = 8.1 Functional
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 60 0 2 1 -1.0 NC(N)=O None
5282379 194984 69 None 25 4 Human 8.2 pIC50 = 8.2 Functional
Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 300 5 1 1 5.6 CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1 None
CHEMBL547 194984 69 None 25 4 Human 8.2 pIC50 = 8.2 Functional
Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Drug Central 300 5 1 1 5.6 CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1 None


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