GPCR CLASS (FAMILY)

Class A (Rhodopsin)

PDB CODE

SPECIES

Homo sapiens

RESOLUTION

2.7 Å

PREFERRED CHAIN

A

REFERENCE

PUBLICATION DATE

Aug. 16, 2017

3D VIEW

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LIGAND INTERACTIONS

LIGANDS

Carazolol - Antagonist pubchem ,

4-carbamoyl-N-[(2R)-2-cyclohexyl-2-phenylacetyl]-L-phenylalanyl-3-bromo-N-methyl-L-phenylalaninamide - Allosteric antagonist pubchem

ENDOGENOUS LIGANDS

noradrenaline, L-NOREPINEPHRINE, (-)-noradrenaline, (-)-adrenaline, Zn2+