GPCR CLASS (FAMILY)
Class A (Rhodopsin)
GPCR SPECIES
Homo sapiens
GPCR PREFERRED CHAIN
R
G PROTEIN (FAMILY)
Gq/11
G PROTEIN SPECIES
Homo sapiens
PDB CODE
RESOLUTION
3.1 Å
REFERENCE
PUBLICATION DATE
Aug. 9, 2023
LIGAND INTERACTIONS
LIGANDS
NTS8–13 - Agonist pubchem ,
SBI-553 - Ago-PAM pubchem gtoplig chembl_ligand
PHYSIOLOGICAL LIGANDS
large neuromedin N (Mouse), neurotensin (Human), neuromedin N (Human), large neuromedin N (Human), large neuromedin N (Rat), large neurotensin (Human), neuromedin N (Mouse)