GPCR CLASS (FAMILY)
Class A (Rhodopsin)
PDB CODE
SPECIES
Homo sapiens
RESOLUTION
3.0 Å
PREFERRED CHAIN
R
PUBLICATION DATE
March 4, 2026
LIGAND INTERACTIONS
LIGANDS
flupentixol - Antagonist pubchem gtoplig chembl_ligand drugbank ,
GEM targeting TM5/6/7 - NAM ,
GEM targeting TM3/4/5 - Unknown ,
GEM targeting TM1/2/4 - Unknown
PHYSIOLOGICAL LIGANDS
5-hydroxytryptamine, noradrenaline, dopamine