Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
AssayType |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
| 2365 | 603 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 603 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 603 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 603 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 603 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 2365 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 2365 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 239 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 4755801 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| CHEMBL297569 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| DB03107 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 603 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 2365 | 603 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 603 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 603 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 603 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 603 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Similar- ity |
Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
Assay Type |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |