|
A2B receptor |
2022-06-19 |
Active |
No
|
AA2BR
|
A2B
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
4UHR |
aa2br_human |
|
CXCR5 |
2022-06-19 |
Inactive |
No
|
CXCR5
|
CXCR5
|
Chemokine |
A (Rhodopsin) |
Human |
CCR7 |
6QZH |
cxcr5_human |
|
5-HT2B receptor |
2022-06-19 |
Intermediate |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
4IB4 |
4ib4 |
|
A2A receptor |
2022-06-20 |
Active |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
3QAK |
3qak |
|
TAS2R8 |
2022-06-19 |
Active |
No
|
TA2R8
|
TAS2R8
|
Taste 2 |
T (Taste 2) |
Human |
D2 receptor |
7JVR |
ta2r8_human |
|
GPR78 |
2022-06-19 |
Active |
No
|
GPR78
|
GPR78
|
A orphans |
A (Rhodopsin) |
Human |
D2 receptor |
7JVR |
gpr78_human |
|
A2A receptor |
2022-06-19 |
Active |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
2YDO |
2ydo |
|
CXCR2 |
2022-06-19 |
Inactive |
Yes
|
CXCR2
|
CXCR2
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
6lfl |
|
CELSR2 |
2022-06-19 |
Intermediate |
No
|
CELR2
|
CELSR2
|
ADGRC |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
celr2_human |
|
TAS2R19 |
2022-06-19 |
Active |
No
|
T2R19
|
TAS2R19
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQG |
t2r19_human |
|
GPR82 |
2022-06-19 |
Intermediate |
No
|
GPR82
|
GPR82
|
A orphans |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
gpr82_human |
|
VPAC1 receptor |
2022-06-19 |
Intermediate |
No
|
VIPR1
|
VPAC1
|
VIP and PACAP |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
vipr1_human |
|
GPR148 |
2022-06-19 |
Inactive |
No
|
GP148
|
GPR148
|
A orphans |
A (Rhodopsin) |
Human |
α1B-adrenoceptor |
7B6W |
gp148_human |
|
M3 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM3
|
M3
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Rat |
M3 receptor |
4U15 |
4u15 |
|
TRH1 receptor |
2022-06-19 |
Inactive |
No
|
TRFR
|
TRH1
|
Thyrotropin-releasing hormone |
A (Rhodopsin) |
Human |
NOP receptor |
5DHG |
trfr_human |
|
A2A receptor |
2022-06-20 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5IU8 |
5iu8 |
|
UT receptor |
2022-06-19 |
Active |
No
|
UR2R
|
UT
|
Urotensin |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
ur2r_human |
|
C5a2 receptor |
2022-06-19 |
Active |
No
|
C5AR2
|
C5a2
|
Complement peptide |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
c5ar2_human |
|
GPR156 |
2022-06-19 |
Intermediate |
No
|
GP156
|
GPR156
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
7CA5 |
gp156_human |
|
GPR50 |
2022-06-19 |
Intermediate |
No
|
MTR1L
|
GPR50
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
mtr1l_human |
|
FZD6 |
2022-06-19 |
Inactive |
No
|
FZD6
|
FZD6
|
Frizzled |
F (Frizzled) |
Human |
FZD5 |
6WW2 |
fzd6_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
4BVN |
4bvn |
|
TAS2R31 |
2022-06-19 |
Inactive |
No
|
T2R31
|
TAS2R31
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQH |
t2r31_human |
|
GPR84 |
2022-06-19 |
Active |
No
|
GPR84
|
GPR84
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6WHA |
gpr84_human |
|
TAS2R5 |
2022-06-19 |
Active |
No
|
TA2R5
|
TAS2R5
|
Taste 2 |
T (Taste 2) |
Human |
CCR1 |
7VL9 |
ta2r5_human |
|
GPR75 |
2022-06-19 |
Inactive |
No
|
GPR75
|
GPR75
|
A orphans |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
gpr75_human |
|
GnRH1 receptor |
2022-06-19 |
Inactive |
Yes
|
GNRHR
|
GnRH1
|
Gonadotrophin-releasing hormone |
A (Rhodopsin) |
Human |
GnRH1 receptor |
7BR3 |
7br3 |
|
LPA4 receptor |
2022-06-19 |
Active |
No
|
LPAR4
|
LPA4
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
κ receptor |
6B73 |
lpar4_human |
|
TAS2R50 |
2022-06-19 |
Active |
No
|
T2R50
|
TAS2R50
|
Taste 2 |
T (Taste 2) |
Human |
D2 receptor |
7JVR |
t2r50_human |
|
GPR55 |
2022-06-19 |
Active |
No
|
GPR55
|
GPR55
|
GPR18, GPR55 and GPR119 |
A (Rhodopsin) |
Human |
AT2 receptor |
5UNG |
gpr55_human |
|
ADGRL3 |
2022-06-19 |
Intermediate |
No
|
AGRL3
|
ADGRL3
|
ADGRL |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrl3_human |
|
CaS receptor |
2022-06-19 |
Active |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7DD7 |
7dd7 |
|
TAS1R1 |
2022-06-19 |
Inactive |
No
|
TS1R1
|
TAS1R1
|
Taste 1 |
C (Glutamate) |
Human |
CaS receptor |
7DD5 |
ts1r1_human |
|
ADGRB1 |
2022-06-19 |
Intermediate |
No
|
AGRB1
|
ADGRB1
|
ADGRB |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrb1_human |
|
CB2 receptor |
2022-06-19 |
Intermediate |
No
|
CNR2
|
CB2
|
Cannabinoid |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
cnr2_human |
|
D1 receptor |
2022-06-19 |
Inactive |
No
|
DRD1
|
D1
|
Dopamine |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
4GBR |
drd1_human |
|
5-HT1B receptor |
2022-06-19 |
Inactive |
Yes
|
5HT1B
|
5-HT1B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAR |
4iar |
|
LPA1 receptor |
2022-06-19 |
Inactive |
Yes
|
LPAR1
|
LPA1
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA1 receptor |
4Z35 |
4z35 |
|
TAS1R1 |
2022-06-19 |
Intermediate |
No
|
TS1R1
|
TAS1R1
|
Taste 1 |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
ts1r1_human |
|
GPR146 |
2022-06-19 |
Intermediate |
No
|
GP146
|
GPR146
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gp146_human |
|
GPR4 |
2022-06-19 |
Active |
No
|
GPR4
|
GPR4
|
A orphans |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
gpr4_human |
|
MRGPRD |
2022-06-19 |
Intermediate |
No
|
MRGRD
|
MRGPRD
|
A orphans |
A (Rhodopsin) |
Human |
CysLT1 receptor |
6RZ4 |
mrgrd_human |
|
GABAB2 |
2022-06-19 |
Active |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
7CA3 |
7ca3 |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
5WKT |
5wkt |
|
D2 receptor |
2022-06-19 |
Inactive |
Yes
|
DRD2
|
D2
|
Dopamine |
A (Rhodopsin) |
Human |
D2 receptor |
6CM4 |
6cm4 |
|
mGlu6 receptor |
2022-06-19 |
Intermediate |
No
|
GRM6
|
mGlu6
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
grm6_human |
|
P2Y12 receptor |
2022-06-19 |
Intermediate |
Yes
|
P2Y12
|
P2Y12
|
P2Y |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
4ntj |
|
CB1 receptor |
2022-06-19 |
Inactive |
Yes
|
CNR1
|
CB1
|
Cannabinoid |
A (Rhodopsin) |
Human |
CB1 receptor |
5TGZ |
5tgz |
|
C5a1 receptor |
2022-06-19 |
Inactive |
Yes
|
C5AR1
|
C5a1
|
Complement peptide |
A (Rhodopsin) |
Human |
C5a1 receptor |
6C1R |
6c1r |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5JTB |
5jtb |
|
P2RY10 |
2022-06-19 |
Intermediate |
No
|
P2Y10
|
P2RY10
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
p2y10_human |
|
SST1 receptor |
2022-06-19 |
Active |
No
|
SSR1
|
SST1
|
Somatostatin |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
ssr1_human |
|
M4 receptor |
2022-06-19 |
Active |
No
|
ACM4
|
M4
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
4MQT |
acm4_human |
|
NPS receptor |
2022-06-19 |
Intermediate |
No
|
NPSR1
|
NPS
|
Neuropeptide S |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
npsr1_human |
|
ADGRF4 |
2022-06-19 |
Active |
No
|
AGRF4
|
ADGRF4
|
ADGRF |
B2 (Adhesion) |
Human |
ADGRF1 |
7WU3 |
agrf4_human |
|
TAS2R38 |
2022-06-19 |
Inactive |
No
|
T2R38
|
TAS2R38
|
Taste 2 |
T (Taste 2) |
Human |
AT1 receptor |
4ZUD |
t2r38_human |
|
OX2 receptor |
2022-06-19 |
Inactive |
Yes
|
OX2R
|
OX2
|
Orexin |
A (Rhodopsin) |
Human |
OX2 receptor |
6TPG |
6tpg |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
3REY |
3rey |
|
5-HT7 receptor |
2022-06-19 |
Active |
No
|
5HT7R
|
5-HT7
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1E receptor |
7E33 |
5ht7r_human |
|
P2RY8 |
2022-06-19 |
Intermediate |
No
|
P2RY8
|
P2RY8
|
A orphans |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
p2ry8_human |
|
TAS2R13 |
2022-06-19 |
Active |
No
|
T2R13
|
TAS2R13
|
Taste 2 |
T (Taste 2) |
Human |
κ receptor |
6B73 |
t2r13_human |
|
GIP receptor |
2022-06-19 |
Inactive |
No
|
GIPR
|
GIP
|
Glucagon |
B1 (Secretin) |
Human |
glucagon receptor |
5YQZ |
gipr_human |
|
GPR88 |
2022-06-19 |
Intermediate |
No
|
GPR88
|
GPR88
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
gpr88_human |
|
chemerin receptor |
2022-06-19 |
Active |
No
|
CML1
|
chemerin
|
Chemerin receptor |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
cml1_human |
|
MT2 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1B
|
MT2
|
Melatonin |
A (Rhodopsin) |
Human |
MT2 receptor |
6ME7 |
6me7 |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
4PXF |
4pxf |
|
TAS2R1 |
2022-06-19 |
Inactive |
No
|
TA2R1
|
TAS2R1
|
Taste 2 |
T (Taste 2) |
Human |
MT1 receptor |
6ME2 |
ta2r1_human |
|
ADGRF2 |
2022-06-19 |
Active |
No
|
AGRF2
|
ADGRF2
|
ADGRF |
B2 (Adhesion) |
Human |
ADGRF1 |
7WU3 |
agrf2_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
7MT9 |
7mt9 |
|
ETB receptor |
2022-06-19 |
Inactive |
Yes
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
5GLH |
5glh |
|
TAS2R30 |
2022-06-19 |
Inactive |
No
|
T2R30
|
TAS2R30
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQH |
t2r30_human |
|
CX3CR1 |
2022-06-19 |
Intermediate |
No
|
CX3C1
|
CX3CR1
|
Chemokine |
A (Rhodopsin) |
Human |
CysLT1 receptor |
6RZ4 |
cx3c1_human |
|
TAS2R46 |
2022-06-19 |
Intermediate |
No
|
T2R46
|
TAS2R46
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
t2r46_human |
|
AT2 receptor |
2022-06-19 |
Active |
Yes
|
AGTR2
|
AT2
|
Angiotensin |
A (Rhodopsin) |
Human |
AT2 receptor |
5XJM |
5xjm |
|
P2Y13 receptor |
2022-06-19 |
Intermediate |
No
|
P2Y13
|
P2Y13
|
P2Y |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
p2y13_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
7VOD |
7vod |
|
ADGRE5 |
2022-06-19 |
Intermediate |
No
|
AGRE5
|
ADGRE5
|
ADGRE |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agre5_human |
|
CELSR1 |
2022-06-19 |
Active |
No
|
CELR1
|
CELSR1
|
ADGRC |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
celr1_human |
|
FZD1 |
2022-06-19 |
Active |
No
|
FZD1
|
FZD1
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd1_human |
|
ADGRE2 |
2022-06-19 |
Active |
No
|
AGRE2
|
ADGRE2
|
ADGRE |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agre2_human |
|
GPR78 |
2022-06-19 |
Intermediate |
No
|
GPR78
|
GPR78
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr78_human |
|
EP1 receptor |
2022-06-19 |
Active |
No
|
PE2R1
|
EP1
|
Prostanoid |
A (Rhodopsin) |
Human |
EP2 receptor |
7CX2 |
pe2r1_human |
|
ADGRB3 |
2022-06-19 |
Active |
No
|
AGRB3
|
ADGRB3
|
ADGRB |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agrb3_human |
|
GPR153 |
2022-06-19 |
Active |
No
|
GP153
|
GPR153
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6WHA |
gp153_human |
|
GPR55 |
2022-06-19 |
Intermediate |
No
|
GPR55
|
GPR55
|
GPR18, GPR55 and GPR119 |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gpr55_human |
|
ADGRE4P |
2022-06-19 |
Inactive |
No
|
AGRE4
|
ADGRE4P
|
ADGRE |
B2 (Adhesion) |
Human |
calcitonin receptor-like receptor |
7KNU |
agre4_human |
|
LPA6 receptor |
2022-06-19 |
Intermediate |
No
|
LPAR6
|
LPA6
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
lpar6_human |
|
NTS2 receptor |
2022-06-19 |
Intermediate |
No
|
NTR2
|
NTS2
|
Neurotensin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
ntr2_human |
|
δ receptor |
2022-06-19 |
Intermediate |
No
|
OPRD
|
δ
|
Opioid |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
oprd_human |
|
A2A receptor |
2022-06-20 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5OM1 |
5om1 |
|
RXFP3 |
2022-06-19 |
Intermediate |
No
|
RL3R1
|
RXFP3
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
rl3r1_human |
|
MRGPRE |
2022-06-19 |
Inactive |
No
|
MRGRE
|
MRGPRE
|
A orphans |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
mrgre_human |
|
BLT2 receptor |
2022-06-19 |
Active |
No
|
LT4R2
|
BLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
BLT1 receptor |
7VKT |
lt4r2_human |
|
GPR171 |
2022-06-19 |
Inactive |
No
|
GP171
|
GPR171
|
A orphans |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
gp171_human |
|
TAS2R39 |
2022-06-19 |
Inactive |
No
|
T2R39
|
TAS2R39
|
Taste 2 |
T (Taste 2) |
Human |
κ receptor |
4DJH |
t2r39_human |
|
5-HT2B receptor |
2022-06-19 |
Intermediate |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
6DRZ |
6drz |
|
PAR3 |
2022-06-19 |
Inactive |
No
|
PAR3
|
PAR3
|
Proteinase-activated |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
par3_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
5A8E |
5a8e |
|
ADGRD1 |
2022-06-19 |
Intermediate |
No
|
AGRD1
|
ADGRD1
|
ADGRD |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrd1_human |
|
FFA1 receptor |
2022-06-19 |
Intermediate |
Yes
|
FFAR1
|
FFA1
|
Free fatty acid |
A (Rhodopsin) |
Human |
FFA1 receptor |
5KW2 |
5kw2 |
|
GPR84 |
2022-06-19 |
Intermediate |
No
|
GPR84
|
GPR84
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr84_human |
|
FPR2/ALX |
2022-06-19 |
Inactive |
No
|
FPR2
|
FPR2/ALX
|
Formylpeptide |
A (Rhodopsin) |
Human |
DP2 receptor |
7M8W |
fpr2_human |
|
ADGRF5 |
2022-06-19 |
Active |
No
|
AGRF5
|
ADGRF5
|
ADGRF |
B2 (Adhesion) |
Human |
ADGRF1 |
7WU3 |
agrf5_human |
|
GPR82 |
2022-06-19 |
Active |
No
|
GPR82
|
GPR82
|
A orphans |
A (Rhodopsin) |
Human |
δ receptor |
6PT2 |
gpr82_human |
|
NTS1 receptor |
2022-06-19 |
Active |
Yes
|
NTR1
|
NTS1
|
Neurotensin |
A (Rhodopsin) |
Rat |
NTS1 receptor |
5T04 |
5t04 |
|
δ receptor |
2022-06-19 |
Active |
Yes
|
OPRD
|
δ
|
Opioid |
A (Rhodopsin) |
Human |
δ receptor |
6PT2 |
6pt2 |
|
oxoglutarate receptor |
2022-06-19 |
Intermediate |
No
|
OXGR1
|
oxoglutarate
|
Oxoglutarate |
A (Rhodopsin) |
Human |
P2Y1 receptor |
4XNW |
oxgr1_human |
|
GPR173 |
2022-06-19 |
Intermediate |
No
|
GP173
|
GPR173
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp173_human |
|
5-HT2C receptor |
2022-06-19 |
Intermediate |
No
|
5HT2C
|
5-HT2C
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht2c_human |
|
A2B receptor |
2022-06-19 |
Inactive |
No
|
AA2BR
|
A2B
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5NM4 |
aa2br_human |
|
TAS2R19 |
2022-06-19 |
Inactive |
No
|
T2R19
|
TAS2R19
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQH |
t2r19_human |
|
MRGPRG |
2022-06-19 |
Active |
No
|
MRGRG
|
MRGPRG
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VDL |
mrgrg_human |
|
GPR82 |
2022-06-19 |
Inactive |
No
|
GPR82
|
GPR82
|
A orphans |
A (Rhodopsin) |
Human |
δ receptor |
4N6H |
gpr82_human |
|
FSH receptor |
2022-06-19 |
Active |
No
|
FSHR
|
FSH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
LH receptor |
7FIG |
fshr_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
5JQH |
5jqh |
|
FZD9 |
2022-06-19 |
Inactive |
No
|
FZD9
|
FZD9
|
Frizzled |
F (Frizzled) |
Human |
FZD4 |
6BD4 |
fzd9_human |
|
α1D-adrenoceptor |
2022-06-19 |
Active |
No
|
ADA1D
|
α1D
|
Adrenoceptors |
A (Rhodopsin) |
Human |
α2B-adrenoceptor |
6K42 |
ada1d_human |
|
GPR12 |
2022-06-19 |
Active |
No
|
GPR12
|
GPR12
|
A orphans |
A (Rhodopsin) |
Human |
LPA1 receptor |
7TD0 |
gpr12_human |
|
mGlu5 receptor |
2022-06-19 |
Intermediate |
Yes
|
GRM5
|
mGlu5
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
6n51 |
|
P2RY10 |
2022-06-19 |
Active |
No
|
P2Y10
|
P2RY10
|
A orphans |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
p2y10_human |
|
GPRC5A |
2022-06-19 |
Inactive |
No
|
RAI3
|
GPRC5A
|
C Orphans |
C (Glutamate) |
Human |
mGlu3 receptor |
7WIH |
rai3_human |
|
TAS2R45 |
2022-06-19 |
Active |
No
|
T2R45
|
TAS2R45
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQG |
t2r45_human |
|
BLT1 receptor |
2022-06-19 |
Inactive |
Yes
|
LT4R1
|
BLT1
|
Leukotriene |
A (Rhodopsin) |
Human |
BLT1 receptor |
7K15 |
7k15 |
|
C3a receptor |
2022-06-19 |
Inactive |
No
|
C3AR
|
C3a
|
Complement peptide |
A (Rhodopsin) |
Human |
C5a1 receptor |
6C1Q |
c3ar_human |
|
TRH1 receptor |
2022-06-19 |
Active |
No
|
TRFR
|
TRH1
|
Thyrotropin-releasing hormone |
A (Rhodopsin) |
Human |
CCK2 receptor |
7F8W |
trfr_human |
|
mGlu2 receptor |
2022-06-19 |
Intermediate |
No
|
GRM2
|
mGlu2
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
grm2_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5UVI |
5uvi |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5IU7 |
5iu7 |
|
GPR26 |
2022-06-19 |
Active |
No
|
GPR26
|
GPR26
|
A orphans |
A (Rhodopsin) |
Human |
D2 receptor |
7JVR |
gpr26_human |
|
GLP-1 receptor |
2022-06-19 |
Active |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
7LCJ |
7lcj |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6FKC |
6fkc |
|
TAS2R3 |
2022-06-19 |
Active |
No
|
TA2R3
|
TAS2R3
|
Taste 2 |
T (Taste 2) |
Human |
GAL1 receptor |
7WQ3 |
ta2r3_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
7WC6 |
7wc6 |
|
TAS2R7 |
2022-06-19 |
Intermediate |
No
|
TA2R7
|
TAS2R7
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
ta2r7_human |
|
TAS2R41 |
2022-06-19 |
Active |
No
|
T2R41
|
TAS2R41
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
7DFL |
t2r41_human |
|
CysLT2 receptor |
2022-06-19 |
Intermediate |
Yes
|
CLTR2
|
CysLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
6rz6 |
|
TAAR2 |
2022-06-19 |
Intermediate |
No
|
TAAR2
|
TAAR2
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar2_human |
|
GPR158 |
2022-06-19 |
Inactive |
Yes
|
GP158
|
GPR158
|
C Orphans |
C (Glutamate) |
Human |
GPR158 |
7SHF |
7shf |
|
GPR135 |
2022-06-19 |
Active |
No
|
GP135
|
GPR135
|
A orphans |
A (Rhodopsin) |
Human |
CCK2 receptor |
7F8W |
gp135_human |
|
5-HT1B receptor |
2022-06-19 |
Inactive |
Yes
|
5HT1B
|
5-HT1B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1B receptor |
7C61 |
7c61 |
|
mGlu5 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM5
|
mGlu5
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N52 |
6n52 |
|
CXCR4 |
2022-06-19 |
Inactive |
Yes
|
CXCR4
|
CXCR4
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR4 |
3ODU |
3odu |
|
GPR35 |
2022-06-19 |
Intermediate |
No
|
GPR35
|
GPR35
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gpr35_human |
|
mGlu1 receptor |
2022-06-19 |
Active |
No
|
GRM1
|
mGlu1
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu2 receptor |
7MTS |
grm1_human |
|
GPR179 |
2022-06-19 |
Active |
No
|
GP179
|
GPR179
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
7C7Q |
gp179_human |
|
TAS2R38 |
2022-06-19 |
Intermediate |
No
|
T2R38
|
TAS2R38
|
Taste 2 |
T (Taste 2) |
Human |
CysLT2 receptor |
6RZ6 |
t2r38_human |
|
TAS2R3 |
2022-06-19 |
Intermediate |
No
|
TA2R3
|
TAS2R3
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
ta2r3_human |
|
FP receptor |
2022-06-19 |
Active |
No
|
PF2R
|
FP
|
Prostanoid |
A (Rhodopsin) |
Human |
EP3 receptor |
6AK3 |
pf2r_human |
|
α1B-adrenoceptor |
2022-06-19 |
Active |
No
|
ADA1B
|
α1B
|
Adrenoceptors |
A (Rhodopsin) |
Human |
α2B-adrenoceptor |
6K42 |
ada1b_human |
|
α2C-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADA2C
|
α2C
|
Adrenoceptors |
A (Rhodopsin) |
Human |
α2C-adrenoceptor |
6KUW |
6kuw |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5IUB |
5iub |
|
CCR6 |
2022-06-19 |
Inactive |
No
|
CCR6
|
CCR6
|
Chemokine |
A (Rhodopsin) |
Human |
CCR7 |
6QZH |
ccr6_human |
|
MCH2 receptor |
2022-06-19 |
Intermediate |
No
|
MCHR2
|
MCH2
|
Melanin-concentrating hormone |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
mchr2_human |
|
LPA3 receptor |
2022-06-19 |
Inactive |
No
|
LPAR3
|
LPA3
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA1 receptor |
4Z35 |
lpar3_human |
|
β1-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
6IBL |
6ibl |
|
P2Y4 receptor |
2022-06-19 |
Inactive |
No
|
P2RY4
|
P2Y4
|
P2Y |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
p2ry4_human |
|
GPR83 |
2022-06-19 |
Inactive |
No
|
GPR83
|
GPR83
|
A orphans |
A (Rhodopsin) |
Human |
Y2 receptor |
7DDZ |
gpr83_human |
|
GAL1 receptor |
2022-06-19 |
Inactive |
No
|
GALR1
|
GAL1
|
Galanin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
galr1_human |
|
CaS receptor |
2022-06-19 |
Inactive |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7E6T |
7e6t |
|
ADGRF3 |
2022-06-19 |
Inactive |
No
|
AGRF3
|
ADGRF3
|
ADGRF |
B2 (Adhesion) |
Human |
calcitonin receptor-like receptor |
7KNU |
agrf3_human |
|
α2C-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADA2C
|
α2C
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
ada2c_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
6PS6 |
6ps6 |
|
OXE receptor |
2022-06-19 |
Intermediate |
No
|
OXER1
|
OXE
|
Leukotriene |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
oxer1_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
2Y02 |
2y02 |
|
GPR87 |
2022-06-19 |
Inactive |
No
|
GPR87
|
GPR87
|
A orphans |
A (Rhodopsin) |
Human |
CXCR4 |
3ODU |
gpr87_human |
|
ADGRF5 |
2022-06-19 |
Intermediate |
No
|
AGRF5
|
ADGRF5
|
ADGRF |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrf5_human |
|
MRGPRX4 |
2022-06-19 |
Intermediate |
No
|
MRGX4
|
MRGPRX4
|
A orphans |
A (Rhodopsin) |
Human |
CysLT1 receptor |
6RZ4 |
mrgx4_human |
|
GPR15 |
2022-06-19 |
Intermediate |
No
|
GPR15
|
GPR15
|
A orphans |
A (Rhodopsin) |
Human |
P2Y1 receptor |
4XNW |
gpr15_human |
|
ADGRG5 |
2022-06-19 |
Inactive |
No
|
AGRG5
|
ADGRG5
|
ADGRG |
B2 (Adhesion) |
Human |
PTH1 receptor |
6FJ3 |
agrg5_human |
|
TAS2R9 |
2022-06-19 |
Inactive |
No
|
TA2R9
|
TAS2R9
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
3RZE |
ta2r9_human |
|
CCR5 |
2022-06-19 |
Inactive |
Yes
|
CCR5
|
CCR5
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
6MEO |
6meo |
|
GPR174 |
2022-06-19 |
Active |
No
|
GP174
|
GPR174
|
A orphans |
A (Rhodopsin) |
Human |
AT2 receptor |
5UNG |
gp174_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
6PS4 |
6ps4 |
|
GPR171 |
2022-06-19 |
Intermediate |
No
|
GP171
|
GPR171
|
A orphans |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
gp171_human |
|
M3 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM3
|
M3
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Rat |
M3 receptor |
4U14 |
4u14 |
|
MT1 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1A
|
MT1
|
Melatonin |
A (Rhodopsin) |
Human |
MT1 receptor |
6ME2 |
6me2 |
|
CaS receptor |
2022-06-19 |
Intermediate |
No
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
casr_human |
|
M3 receptor |
2022-06-19 |
Inactive |
No
|
ACM3
|
M3
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M3 receptor |
5ZHP |
acm3_human |
|
β3-adrenoceptor |
2022-06-20 |
Active |
No
|
ADRB3
|
β3
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β3-adrenoceptor |
7DH5 |
adrb3_human |
|
CCR9 |
2022-06-19 |
Active |
No
|
CCR9
|
CCR9
|
Chemokine |
A (Rhodopsin) |
Human |
CCR6 |
6WWZ |
ccr9_human |
|
GPR176 |
2022-06-19 |
Intermediate |
No
|
GP176
|
GPR176
|
A orphans |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
gp176_human |
|
LGR5 |
2022-06-19 |
Inactive |
No
|
LGR5
|
LGR5
|
A orphans |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
lgr5_human |
|
NPS receptor |
2022-06-19 |
Active |
No
|
NPSR1
|
NPS
|
Neuropeptide S |
A (Rhodopsin) |
Human |
OT receptor |
7RYC |
npsr1_human |
|
ADGRD2 |
2022-06-19 |
Active |
No
|
AGRD2
|
ADGRD2
|
ADGRD |
B2 (Adhesion) |
Human |
ADGRD1 |
7WU2 |
agrd2_human |
|
LGR4 |
2022-06-19 |
Inactive |
No
|
LGR4
|
LGR4
|
A orphans |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
lgr4_human |
|
BB3 receptor |
2022-06-19 |
Intermediate |
No
|
BRS3
|
BB3
|
Bombesin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
brs3_human |
|
ADGRV1 |
2022-06-19 |
Intermediate |
No
|
AGRV1
|
ADGRV1
|
ADGRV |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrv1_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5NM4 |
5nm4 |
|
NK2 receptor |
2022-06-19 |
Inactive |
No
|
NK2R
|
NK2
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
6HLP |
nk2r_human |
|
MT2 receptor |
2022-06-19 |
Intermediate |
No
|
MTR1B
|
MT2
|
Melatonin |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
mtr1b_human |
|
HCA2 receptor |
2022-06-19 |
Intermediate |
No
|
HCAR2
|
HCA2
|
Hydroxycarboxylic acid |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
hcar2_human |
|
CCR5 |
2022-06-19 |
Inactive |
Yes
|
CCR5
|
CCR5
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
6AKX |
6akx |
|
HCA2 receptor |
2022-06-19 |
Inactive |
No
|
HCAR2
|
HCA2
|
Hydroxycarboxylic acid |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
hcar2_human |
|
CXCR1 |
2022-06-19 |
Active |
No
|
CXCR1
|
CXCR1
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFO |
cxcr1_human |
|
CELSR1 |
2022-06-19 |
Intermediate |
No
|
CELR1
|
CELSR1
|
ADGRC |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
celr1_human |
|
succinate receptor |
2022-06-19 |
Intermediate |
Yes
|
SUCR1
|
succinate
|
Succinate |
A (Rhodopsin) |
Rat |
succinate receptor |
6RNK |
6rnk |
|
LPA5 receptor |
2022-06-20 |
Intermediate |
No
|
LPAR5
|
LPA5
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
lpar5_human |
|
CCR3 |
2022-06-19 |
Inactive |
No
|
CCR3
|
CCR3
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ccr3_human |
|
NK1 receptor |
2022-06-19 |
Inactive |
Yes
|
NK1R
|
NK1
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
6HLO |
6hlo |
|
SMO |
2022-06-20 |
Inactive |
Yes
|
SMO
|
SMO
|
Frizzled |
F (Frizzled) |
Human |
SMO |
4QIN |
4qin |
|
TAS2R16 |
2022-06-19 |
Intermediate |
No
|
T2R16
|
TAS2R16
|
Taste 2 |
T (Taste 2) |
Human |
P2Y1 receptor |
4XNW |
t2r16_human |
|
C5a1 receptor |
2022-06-19 |
Intermediate |
No
|
C5AR1
|
C5a1
|
Complement peptide |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
c5ar1_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TOD |
6tod |
|
TA1 receptor |
2022-06-19 |
Intermediate |
No
|
TAAR1
|
TA1
|
Trace amine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar1_human |
|
RXFP2 |
2022-06-19 |
Inactive |
No
|
RXFP2
|
RXFP2
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
rxfp2_human |
|
LPA3 receptor |
2022-06-19 |
Active |
No
|
LPAR3
|
LPA3
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA1 receptor |
7TD0 |
lpar3_human |
|
GLP-1 receptor |
2021-11-02 |
Intermediate |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
5nx2 |
|
FFA1 receptor |
2022-06-19 |
Active |
No
|
FFAR1
|
FFA1
|
Free fatty acid |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
ffar1_human |
|
GPR19 |
2022-06-19 |
Active |
No
|
GPR19
|
GPR19
|
A orphans |
A (Rhodopsin) |
Human |
CCK1 receptor |
7EZM |
gpr19_human |
|
GPR4 |
2022-06-19 |
Inactive |
No
|
GPR4
|
GPR4
|
A orphans |
A (Rhodopsin) |
Human |
CCR2 |
5T1A |
gpr4_human |
|
CCR3 |
2022-06-19 |
Active |
No
|
CCR3
|
CCR3
|
Chemokine |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
ccr3_human |
|
D2 receptor |
2022-06-19 |
Intermediate |
No
|
DRD2
|
D2
|
Dopamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
drd2_human |
|
TP receptor |
2022-06-19 |
Inactive |
No
|
TA2R
|
TP
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
ta2r_human |
|
CaS receptor |
2022-06-19 |
Active |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7DD6 |
7dd6 |
|
GPRC5D |
2022-06-19 |
Intermediate |
No
|
GPC5D
|
GPRC5D
|
C Orphans |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
gpc5d_human |
|
mGlu3 receptor |
2022-06-19 |
Active |
No
|
GRM3
|
mGlu3
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu2 receptor |
7MTS |
grm3_human |
|
CB2 receptor |
2022-06-19 |
Inactive |
Yes
|
CNR2
|
CB2
|
Cannabinoid |
A (Rhodopsin) |
Human |
CB2 receptor |
5ZTY |
5zty |
|
TP receptor |
2022-06-19 |
Intermediate |
Yes
|
TA2R
|
TP
|
Prostanoid |
A (Rhodopsin) |
Human |
TP receptor |
6IIV |
6iiv |
|
M2 receptor |
2022-06-19 |
Active |
Yes
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
4MQT |
4mqt |
|
mGlu6 receptor |
2022-06-19 |
Active |
No
|
GRM6
|
mGlu6
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu4 receptor |
7E9H |
grm6_human |
|
GPR119 |
2022-06-19 |
Inactive |
No
|
GP119
|
GPR119
|
GPR18, GPR55 and GPR119 |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
gp119_human |
|
GPR61 |
2022-06-19 |
Intermediate |
No
|
GPR61
|
GPR61
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr61_human |
|
OPN4 |
2022-06-19 |
Inactive |
No
|
OPN4
|
OPN4
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
6I9K |
opn4_human |
|
PAF receptor |
2022-06-19 |
Inactive |
No
|
PTAFR
|
PAF
|
Platelet-activating factor |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ptafr_human |
|
GPR39 |
2022-06-19 |
Inactive |
No
|
GPR39
|
GPR39
|
A orphans |
A (Rhodopsin) |
Human |
NTS1 receptor |
6YVR |
gpr39_human |
|
FFA2 receptor |
2022-06-19 |
Inactive |
No
|
FFAR2
|
FFA2
|
Free fatty acid |
A (Rhodopsin) |
Human |
CCK1 receptor |
7F8Y |
ffar2_human |
|
FFA2 receptor |
2022-06-19 |
Active |
No
|
FFAR2
|
FFA2
|
Free fatty acid |
A (Rhodopsin) |
Human |
GAL1 receptor |
7WQ3 |
ffar2_human |
|
TAS2R16 |
2022-06-19 |
Active |
No
|
T2R16
|
TAS2R16
|
Taste 2 |
T (Taste 2) |
Human |
CCR1 |
7VL9 |
t2r16_human |
|
5-HT1F receptor |
2022-06-19 |
Intermediate |
No
|
5HT1F
|
5-HT1F
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht1f_human |
|
GPR85 |
2022-06-19 |
Intermediate |
No
|
GPR85
|
GPR85
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr85_human |
|
TAS1R1 |
2022-06-19 |
Active |
No
|
TS1R1
|
TAS1R1
|
Taste 1 |
C (Glutamate) |
Human |
CaS receptor |
7DD6 |
ts1r1_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
3NY8 |
3ny8 |
|
GPR45 |
2022-06-19 |
Intermediate |
No
|
GPR45
|
GPR45
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr45_human |
|
PAC1 receptor |
2022-06-19 |
Intermediate |
No
|
PACR
|
PAC1
|
VIP and PACAP |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
pacr_human |
|
GPRC5B |
2022-06-19 |
Inactive |
No
|
GPC5B
|
GPRC5B
|
C Orphans |
C (Glutamate) |
Human |
mGlu3 receptor |
7WIH |
gpc5b_human |
|
GPR31 |
2022-06-19 |
Intermediate |
No
|
GPR31
|
GPR31
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gpr31_human |
|
GPR62 |
2022-06-19 |
Inactive |
No
|
GPR62
|
GPR62
|
A orphans |
A (Rhodopsin) |
Human |
D3 receptor |
3PBL |
gpr62_human |
|
δ receptor |
2022-06-19 |
Inactive |
Yes
|
OPRD
|
δ
|
Opioid |
A (Rhodopsin) |
Human |
δ receptor |
4RWD |
4rwd |
|
TSH receptor |
2022-06-19 |
Active |
No
|
TSHR
|
TSH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
LH receptor |
7FIG |
tshr_human |
|
GPR20 |
2022-06-19 |
Active |
No
|
GPR20
|
GPR20
|
A orphans |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
gpr20_human |
|
ghrelin receptor |
2022-06-19 |
Intermediate |
No
|
GHSR
|
ghrelin
|
Ghrelin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
ghsr_human |
|
XCR1 |
2022-06-19 |
Intermediate |
No
|
XCR1
|
XCR1
|
Chemokine |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
xcr1_human |
|
TAAR3 |
2022-06-19 |
Active |
No
|
TAAR3
|
TAAR3
|
A orphans |
A (Rhodopsin) |
Human |
α2A-adrenoceptor |
7EJ8 |
taar3_human |
|
5-HT2B receptor |
2022-06-19 |
Intermediate |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
4NC3 |
4nc3 |
|
GPR85 |
2022-06-19 |
Active |
No
|
GPR85
|
GPR85
|
A orphans |
A (Rhodopsin) |
Human |
D1 receptor |
7JVQ |
gpr85_human |
|
ADGRF3 |
2022-06-19 |
Active |
No
|
AGRF3
|
ADGRF3
|
ADGRF |
B2 (Adhesion) |
Human |
ADGRF1 |
7WU3 |
agrf3_human |
|
V1A receptor |
2022-06-19 |
Intermediate |
No
|
V1AR
|
V1A
|
Vasopressin and oxytocin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
v1ar_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
4ZJ8 |
4zj8 |
|
α2C-adrenoceptor |
2022-06-19 |
Active |
No
|
ADA2C
|
α2C
|
Adrenoceptors |
A (Rhodopsin) |
Human |
α2A-adrenoceptor |
7EJ8 |
ada2c_human |
|
GPRC5C |
2022-06-19 |
Intermediate |
No
|
GPC5C
|
GPRC5C
|
C Orphans |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
gpc5c_human |
|
NPFF1 receptor |
2022-06-19 |
Inactive |
No
|
NPFF1
|
NPFF1
|
Neuropeptide FF/neuropeptide AF |
A (Rhodopsin) |
Human |
OX1 receptor |
6TO7 |
npff1_human |
|
CELSR3 |
2022-06-19 |
Active |
No
|
CELR3
|
CELSR3
|
ADGRC |
B2 (Adhesion) |
Human |
ADGRD1 |
7WU2 |
celr3_human |
|
TAAR6 |
2022-06-19 |
Active |
No
|
TAAR6
|
TAAR6
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1F receptor |
7EXD |
taar6_human |
|
PTH2 receptor |
2022-06-19 |
Intermediate |
No
|
PTH2R
|
PTH2
|
Parathyroid hormone |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
pth2r_human |
|
MC4 receptor |
2022-06-19 |
Intermediate |
Yes
|
MC4R
|
MC4
|
Melanocortin |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
6w25 |
|
5-HT1B receptor |
2022-06-19 |
Inactive |
Yes
|
5HT1B
|
5-HT1B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAQ |
4iaq |
|
GPR162 |
2022-06-19 |
Active |
No
|
GP162
|
GPR162
|
A orphans |
A (Rhodopsin) |
Human |
D2 receptor |
7JVR |
gp162_human |
|
OPN1SW |
2022-06-19 |
Intermediate |
No
|
OPSB
|
OPN1SW
|
Opsins |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
opsb_human |
|
GPR21 |
2022-06-19 |
Active |
No
|
GPR21
|
GPR21
|
A orphans |
A (Rhodopsin) |
Human |
GPR52 |
6LI3 |
gpr21_human |
|
EP1 receptor |
2022-06-19 |
Inactive |
No
|
PE2R1
|
EP1
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
pe2r1_human |
|
SMO |
2022-06-19 |
Inactive |
Yes
|
SMO
|
SMO
|
Frizzled |
F (Frizzled) |
Human |
SMO |
5V56 |
5v56 |
|
mGlu4 receptor |
2022-06-19 |
Intermediate |
No
|
GRM4
|
mGlu4
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
grm4_human |
|
GABAB2 |
2022-06-19 |
Intermediate |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
7CA5 |
7ca5 |
|
M2 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
5ZKC |
5zkc |
|
CCR4 |
2022-06-19 |
Inactive |
No
|
CCR4
|
CCR4
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ccr4_human |
|
GPR42 |
2022-06-19 |
Intermediate |
No
|
GPR42
|
GPR42
|
Free fatty acid |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
gpr42_human |
|
PAR1 |
2022-06-19 |
Active |
No
|
PAR1
|
PAR1
|
Proteinase-activated |
A (Rhodopsin) |
Human |
κ receptor |
6B73 |
par1_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TQ6 |
6tq6 |
|
NPBW1 receptor |
2022-06-19 |
Active |
No
|
NPBW1
|
NPBW1
|
Neuropeptide W/neuropeptide B |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
npbw1_human |
|
CELSR3 |
2022-06-19 |
Intermediate |
No
|
CELR3
|
CELSR3
|
ADGRC |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
celr3_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
5W0P |
5w0p |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
4J4Q |
4j4q |
|
ADGRV1 |
2022-06-19 |
Active |
No
|
AGRV1
|
ADGRV1
|
ADGRV |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agrv1_human |
|
GPR45 |
2022-06-19 |
Inactive |
No
|
GPR45
|
GPR45
|
A orphans |
A (Rhodopsin) |
Human |
D2 receptor |
6LUQ |
gpr45_human |
|
GPR3 |
2022-06-19 |
Inactive |
No
|
GPR3
|
GPR3
|
A orphans |
A (Rhodopsin) |
Human |
LPA1 receptor |
4Z35 |
gpr3_human |
|
P2Y12 receptor |
2022-06-20 |
Intermediate |
Yes
|
P2Y12
|
P2Y12
|
P2Y |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4PY0 |
4py0 |
|
GPR33 |
2022-06-19 |
Inactive |
No
|
GPR33
|
GPR33
|
A orphans |
A (Rhodopsin) |
Human |
DP2 receptor |
7M8W |
gpr33_human |
|
TAS2R10 |
2022-06-19 |
Inactive |
No
|
T2R10
|
TAS2R10
|
Taste 2 |
T (Taste 2) |
Human |
α1B-adrenoceptor |
7B6W |
t2r10_human |
|
GPR15 |
2022-06-19 |
Inactive |
No
|
GPR15
|
GPR15
|
A orphans |
A (Rhodopsin) |
Human |
apelin receptor |
5VBL |
gpr15_human |
|
FPR1 |
2022-06-19 |
Inactive |
No
|
FPR1
|
FPR1
|
Formylpeptide |
A (Rhodopsin) |
Human |
DP2 receptor |
7M8W |
fpr1_human |
|
5-HT1A receptor |
2022-06-19 |
Intermediate |
No
|
5HT1A
|
5-HT1A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht1a_human |
|
MAS1 |
2022-06-19 |
Active |
No
|
MAS
|
MAS1
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VDL |
mas_human |
|
δ receptor |
2022-06-19 |
Inactive |
Yes
|
OPRD
|
δ
|
Opioid |
A (Rhodopsin) |
Human |
δ receptor |
4N6H |
4n6h |
|
TSH receptor |
2022-06-19 |
Inactive |
No
|
TSHR
|
TSH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
tshr_human |
|
ADGRA1 |
2022-06-19 |
Active |
No
|
AGRA1
|
ADGRA1
|
ADGRA |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agra1_human |
|
D4 receptor |
2022-06-19 |
Active |
No
|
DRD4
|
D4
|
Dopamine |
A (Rhodopsin) |
Human |
D3 receptor |
7CMV |
drd4_human |
|
GPR39 |
2022-06-19 |
Active |
No
|
GPR39
|
GPR39
|
A orphans |
A (Rhodopsin) |
Human |
NTS1 receptor |
4XES |
gpr39_human |
|
DP1 receptor |
2022-06-19 |
Intermediate |
No
|
PD2R
|
DP1
|
Prostanoid |
A (Rhodopsin) |
Human |
TP receptor |
6IIV |
pd2r_human |
|
MRGPRG |
2022-06-19 |
Intermediate |
No
|
MRGRG
|
MRGPRG
|
A orphans |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ6 |
mrgrg_human |
|
OPN1SW |
2022-06-19 |
Active |
No
|
OPSB
|
OPN1SW
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
4X1H |
opsb_human |
|
FZD4 |
2022-06-19 |
Active |
No
|
FZD4
|
FZD4
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd4_human |
|
AT2 receptor |
2022-06-19 |
Active |
Yes
|
AGTR2
|
AT2
|
Angiotensin |
A (Rhodopsin) |
Human |
AT2 receptor |
7C6A |
7c6a |
|
CaS receptor |
2022-06-19 |
Inactive |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7DTT |
7dtt |
|
H3 receptor |
2022-06-19 |
Active |
No
|
HRH3
|
H3
|
Histamine |
A (Rhodopsin) |
Human |
H1 receptor |
7DFL |
hrh3_human |
|
GnRH1 receptor |
2022-06-19 |
Intermediate |
No
|
GNRHR
|
GnRH1
|
Gonadotrophin-releasing hormone |
A (Rhodopsin) |
Human |
PAR1 |
3VW7 |
gnrhr_human |
|
FFA1 receptor |
2022-06-19 |
Intermediate |
Yes
|
FFAR1
|
FFA1
|
Free fatty acid |
A (Rhodopsin) |
Human |
FFA1 receptor |
5TZY |
5tzy |
|
DP1 receptor |
2022-06-19 |
Active |
No
|
PD2R
|
DP1
|
Prostanoid |
A (Rhodopsin) |
Human |
EP2 receptor |
7CX2 |
pd2r_human |
|
ADGRB3 |
2022-06-19 |
Inactive |
No
|
AGRB3
|
ADGRB3
|
ADGRB |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrb3_human |
|
MRGPRD |
2022-06-19 |
Active |
No
|
MRGRD
|
MRGPRD
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VDL |
mrgrd_human |
|
SST4 receptor |
2022-06-19 |
Inactive |
No
|
SSR4
|
SST4
|
Somatostatin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
ssr4_human |
|
OX2 receptor |
2022-06-19 |
Inactive |
Yes
|
OX2R
|
OX2
|
Orexin |
A (Rhodopsin) |
Human |
OX2 receptor |
6TPN |
6tpn |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6FK6 |
6fk6 |
|
GABAB1 |
2022-06-19 |
Intermediate |
No
|
GABR1
|
GABAB1
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
7CA5 |
gabr1_human |
|
A1 receptor |
2022-06-19 |
Inactive |
Yes
|
AA1R
|
A1
|
Adenosine |
A (Rhodopsin) |
Human |
A1 receptor |
5N2S |
5n2s |
|
GPR161 |
2022-06-19 |
Intermediate |
No
|
GP161
|
GPR161
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp161_human |
|
CRF1 receptor |
2022-06-20 |
Inactive |
Yes
|
CRFR1
|
CRF1
|
Corticotropin-releasing factor |
B1 (Secretin) |
Human |
CRF1 receptor |
4K5Y |
4k5y |
|
MRGPRX2 |
2022-06-19 |
Active |
Yes
|
MRGX2
|
MRGPRX2
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VV0 |
7vv0 |
|
TAS2R20 |
2022-06-19 |
Inactive |
No
|
T2R20
|
TAS2R20
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQH |
t2r20_human |
|
GPR61 |
2022-06-19 |
Active |
No
|
GPR61
|
GPR61
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1E receptor |
7E33 |
gpr61_human |
|
α1D-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADA1D
|
α1D
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
ada1d_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
7WC9 |
7wc9 |
|
VPAC2 receptor |
2022-06-19 |
Intermediate |
No
|
VIPR2
|
VPAC2
|
VIP and PACAP |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
vipr2_human |
|
5-HT2B receptor |
2022-06-19 |
Intermediate |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
6DRY |
6dry |
|
GPR65 |
2022-06-19 |
Intermediate |
No
|
PSYR
|
GPR65
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
psyr_human |
|
MRGPRD |
2022-06-19 |
Inactive |
No
|
MRGRD
|
MRGPRD
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
mrgrd_human |
|
AT2 receptor |
2022-06-19 |
Active |
Yes
|
AGTR2
|
AT2
|
Angiotensin |
A (Rhodopsin) |
Human |
AT2 receptor |
7JNI |
7jni |
|
LGR4 |
2022-06-19 |
Intermediate |
No
|
LGR4
|
LGR4
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
lgr4_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
5TE3 |
5te3 |
|
TAAR9 |
2022-06-19 |
Intermediate |
No
|
TAAR9
|
TAAR9
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar9_human |
|
ADGRB1 |
2022-06-19 |
Inactive |
No
|
AGRB1
|
ADGRB1
|
ADGRB |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrb1_human |
|
MT2 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1B
|
MT2
|
Melatonin |
A (Rhodopsin) |
Human |
MT2 receptor |
6ME9 |
6me9 |
|
ADGRF1 |
2022-06-19 |
Intermediate |
No
|
AGRF1
|
ADGRF1
|
ADGRF |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrf1_human |
|
S1P4 receptor |
2022-06-19 |
Inactive |
No
|
S1PR4
|
S1P4
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
s1pr4_human |
|
TAAR3 |
2022-06-19 |
Intermediate |
No
|
TAAR3
|
TAAR3
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar3_human |
|
TAAR8 |
2022-06-19 |
Intermediate |
No
|
TAAR8
|
TAAR8
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar8_human |
|
GPR152 |
2022-06-19 |
Active |
No
|
GP152
|
GPR152
|
A orphans |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
gp152_human |
|
CCR2 |
2022-06-19 |
Inactive |
Yes
|
CCR2
|
CCR2
|
Chemokine |
A (Rhodopsin) |
Human |
CCR2 |
6GPS |
6gps |
|
GPR6 |
2022-06-19 |
Inactive |
No
|
GPR6
|
GPR6
|
A orphans |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
gpr6_human |
|
LPA6 receptor |
2022-06-19 |
Inactive |
No
|
LPAR6
|
LPA6
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
lpar6_human |
|
Olfactory receptor 1G1 |
2022-06-19 |
Active |
No
|
OR1G1
|
Olfactory 1G1
|
Olfactory |
A (Rhodopsin) |
Human |
LPA1 receptor |
7TD0 |
or1g1_human |
|
GIP receptor |
2022-06-19 |
Intermediate |
No
|
GIPR
|
GIP
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
gipr_human |
|
C3a receptor |
2022-06-19 |
Active |
No
|
C3AR
|
C3a
|
Complement peptide |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
c3ar_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5IUA |
5iua |
|
GPR141 |
2022-06-19 |
Active |
No
|
GP141
|
GPR141
|
A orphans |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
gp141_human |
|
FZD5 |
2022-06-19 |
Active |
No
|
FZD5
|
FZD5
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd5_human |
|
OPN1SW |
2022-06-20 |
Inactive |
No
|
OPSB
|
OPN1SW
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
1U19 |
opsb_human |
|
NK3 receptor |
2022-06-19 |
Inactive |
No
|
NK3R
|
NK3
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
6HLP |
nk3r_human |
|
ADGRA2 |
2022-06-19 |
Active |
No
|
AGRA2
|
ADGRA2
|
ADGRA |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agra2_human |
|
Olfactory receptor 1A1 |
2022-06-19 |
Inactive |
No
|
OR1A1
|
Olfactory 1A1
|
Olfactory |
A (Rhodopsin) |
Human |
A1 receptor |
5UEN |
or1a1_human |
|
GLP-1 receptor |
2022-06-19 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
6LN2 |
6ln2 |
|
TAS2R40 |
2022-06-19 |
Active |
No
|
T2R40
|
TAS2R40
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQG |
t2r40_human |
|
kisspeptin receptor |
2022-06-19 |
Inactive |
No
|
KISSR
|
kisspeptin
|
Kisspeptin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
kissr_human |
|
TAS2R60 |
2022-06-19 |
Active |
No
|
T2R60
|
TAS2R60
|
Taste 2 |
T (Taste 2) |
Human |
κ receptor |
6B73 |
t2r60_human |
|
GPR50 |
2022-06-19 |
Inactive |
No
|
MTR1L
|
GPR50
|
A orphans |
A (Rhodopsin) |
Human |
MT1 receptor |
6ME2 |
mtr1l_human |
|
A2A receptor |
2022-06-19 |
Active |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5WF6 |
5wf6 |
|
CCK1 receptor |
2022-06-19 |
Inactive |
Yes
|
CCKAR
|
CCK1
|
Cholecystokinin |
A (Rhodopsin) |
Human |
CCK1 receptor |
7F8U |
7f8u |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
5EN0 |
5en0 |
|
CCRL2 |
2022-06-19 |
Active |
No
|
CCRL2
|
CCRL2
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
7O7F |
ccrl2_human |
|
LPA6 receptor |
2022-06-19 |
Intermediate |
Yes
|
Q08BG4
|
LPA6
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Zebrafish |
LPA6 receptor |
5XSZ |
5xsz |
|
β2-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
4LDO |
4ldo |
|
oxoglutarate receptor |
2022-06-19 |
Inactive |
No
|
OXGR1
|
oxoglutarate
|
Oxoglutarate |
A (Rhodopsin) |
Human |
CCR7 |
6QZH |
oxgr1_human |
|
P2Y2 receptor |
2022-06-19 |
Inactive |
No
|
P2RY2
|
P2Y2
|
P2Y |
A (Rhodopsin) |
Human |
μ receptor |
4DKL |
p2ry2_human |
|
ADGRG1 |
2022-06-19 |
Intermediate |
No
|
AGRG1
|
ADGRG1
|
ADGRG |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrg1_human |
|
FFA4 receptor |
2022-06-19 |
Inactive |
No
|
FFAR4
|
FFA4
|
Free fatty acid |
A (Rhodopsin) |
Human |
OX2 receptor |
5WQC |
ffar4_human |
|
MC2 receptor |
2022-06-19 |
Inactive |
No
|
ACTHR
|
MC2
|
Melanocortin |
A (Rhodopsin) |
Human |
CB1 receptor |
5TGZ |
acthr_human |
|
TAS2R14 |
2022-06-19 |
Intermediate |
No
|
T2R14
|
TAS2R14
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
t2r14_human |
|
TAS2R46 |
2022-06-19 |
Inactive |
No
|
T2R46
|
TAS2R46
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQH |
t2r46_human |
|
CCRL2 |
2022-06-19 |
Intermediate |
No
|
CCRL2
|
CCRL2
|
Chemokine |
A (Rhodopsin) |
Human |
PAR1 |
3VW7 |
ccrl2_human |
|
P2Y11 receptor |
2022-06-19 |
Inactive |
No
|
P2Y11
|
P2Y11
|
P2Y |
A (Rhodopsin) |
Human |
apelin receptor |
5VBL |
p2y11_human |
|
PAR4 |
2022-06-19 |
Intermediate |
No
|
PAR4
|
PAR4
|
Proteinase-activated |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
par4_human |
|
OX2 receptor |
2022-06-19 |
Inactive |
Yes
|
OX2R
|
OX2
|
Orexin |
A (Rhodopsin) |
Human |
OX2 receptor |
6TPJ |
6tpj |
|
QRFP receptor |
2022-06-19 |
Active |
No
|
QRFPR
|
QRFP
|
Peptide P518 |
A (Rhodopsin) |
Human |
OX2 receptor |
7L1V |
qrfpr_human |
|
β1-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BU6 |
7bu6 |
|
5-HT2A receptor |
2022-06-20 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
7WC8 |
7wc8 |
|
GPR62 |
2022-06-19 |
Intermediate |
No
|
GPR62
|
GPR62
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr62_human |
|
SST1 receptor |
2022-06-19 |
Intermediate |
No
|
SSR1
|
SST1
|
Somatostatin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
ssr1_human |
|
FZD10 |
2022-06-19 |
Inactive |
No
|
FZD10
|
FZD10
|
Frizzled |
F (Frizzled) |
Human |
FZD4 |
6BD4 |
fzd10_human |
|
SST5 receptor |
2022-06-19 |
Inactive |
No
|
SSR5
|
SST5
|
Somatostatin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
ssr5_human |
|
GPR158 |
2022-06-19 |
Inactive |
Yes
|
GP158
|
GPR158
|
C Orphans |
C (Glutamate) |
Human |
GPR158 |
7EWP |
7ewp |
|
ETB receptor |
2022-06-19 |
Inactive |
Yes
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
6IGL |
6igl |
|
M5 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM5
|
M5
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M5 receptor |
6OL9 |
6ol9 |
|
ADGRG5 |
2022-06-19 |
Active |
No
|
AGRG5
|
ADGRG5
|
ADGRG |
B2 (Adhesion) |
Human |
ADGRG1 |
7SF8 |
agrg5_human |
|
GABAB2 |
2022-06-19 |
Inactive |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
6WIV |
6wiv |
|
M2 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
3UON |
3uon |
|
ADGRG6 |
2022-06-19 |
Active |
No
|
AGRG6
|
ADGRG6
|
ADGRG |
B2 (Adhesion) |
Human |
ADGRG4 |
7WUJ |
agrg6_human |
|
TAAR5 |
2022-06-19 |
Intermediate |
No
|
TAAR5
|
TAAR5
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar5_human |
|
Olfactory receptor 1A1 |
2022-06-19 |
Active |
No
|
OR1A1
|
Olfactory 1A1
|
Olfactory |
A (Rhodopsin) |
Human |
A1 receptor |
6D9H |
or1a1_human |
|
β2-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
4LDE |
4lde |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TQ7 |
6tq7 |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6A94 |
6a94 |
|
TAS2R41 |
2022-06-19 |
Inactive |
No
|
T2R41
|
TAS2R41
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
3RZE |
t2r41_human |
|
Y2 receptor |
2022-06-19 |
Active |
No
|
NPY2R
|
Y2
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
OX2 receptor |
7L1V |
npy2r_human |
|
OPN3 |
2022-06-19 |
Active |
No
|
OPN3
|
OPN3
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
4X1H |
opn3_human |
|
MT1 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1A
|
MT1
|
Melatonin |
A (Rhodopsin) |
Human |
MT1 receptor |
6ME4 |
6me4 |
|
GPR87 |
2022-06-19 |
Intermediate |
No
|
GPR87
|
GPR87
|
A orphans |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
gpr87_human |
|
P2Y14 receptor |
2022-06-19 |
Intermediate |
No
|
P2Y14
|
P2Y14
|
P2Y |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
p2y14_human |
|
PAR1 |
2022-06-19 |
Intermediate |
Yes
|
PAR1
|
PAR1
|
Proteinase-activated |
A (Rhodopsin) |
Human |
PAR1 |
3VW7 |
3vw7 |
|
α2A-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADA2A
|
α2A
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
ada2a_human |
|
M2 receptor |
2022-06-19 |
Active |
Yes
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
6U1N |
6u1n |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6GT3 |
6gt3 |
|
S1P5 receptor |
2022-06-19 |
Intermediate |
No
|
S1PR5
|
S1P5
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
s1pr5_human |
|
ADGRL4 |
2022-06-19 |
Inactive |
No
|
AGRL4
|
ADGRL4
|
ADGRL |
B2 (Adhesion) |
Human |
calcitonin receptor-like receptor |
7KNU |
agrl4_human |
|
DP2 receptor |
2022-06-19 |
Inactive |
Yes
|
PD2R2
|
DP2
|
Prostanoid |
A (Rhodopsin) |
Human |
DP2 receptor |
6D26 |
6d26 |
|
IP receptor |
2022-06-19 |
Inactive |
No
|
PI2R
|
IP
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
pi2r_human |
|
ADGRA2 |
2022-06-19 |
Inactive |
No
|
AGRA2
|
ADGRA2
|
ADGRA |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agra2_human |
|
LPA6 receptor |
2022-06-19 |
Active |
No
|
LPAR6
|
LPA6
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
lpar6_human |
|
AT1 receptor |
2022-06-19 |
Inactive |
Yes
|
AGTR1
|
AT1
|
Angiotensin |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
4zud |
|
LPA2 receptor |
2022-06-19 |
Intermediate |
No
|
LPAR2
|
LPA2
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
lpar2_human |
|
GLP-1 receptor |
2022-06-19 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
6KJV |
6kjv |
|
α1A-adrenoceptor |
2022-06-19 |
Active |
No
|
ADA1A
|
α1A
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BU7 |
ada1a_human |
|
C5a1 receptor |
2022-06-19 |
Inactive |
Yes
|
C5AR1
|
C5a1
|
Complement peptide |
A (Rhodopsin) |
Human |
C5a1 receptor |
5O9H |
5o9h |
|
NTS2 receptor |
2022-06-19 |
Inactive |
No
|
NTR2
|
NTS2
|
Neurotensin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6YVR |
ntr2_human |
|
GPR87 |
2022-06-19 |
Active |
No
|
GPR87
|
GPR87
|
A orphans |
A (Rhodopsin) |
Human |
B2 receptor |
7F2O |
gpr87_human |
|
GPRC6 receptor |
2022-06-19 |
Intermediate |
No
|
GPC6A
|
GPRC6
|
C Orphans |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
gpc6a_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6MH8 |
6mh8 |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6JZH |
6jzh |
|
LPA1 receptor |
2022-06-19 |
Inactive |
Yes
|
LPAR1
|
LPA1
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA1 receptor |
4Z36 |
4z36 |
|
Rhodopsin |
2022-06-19 |
Intermediate |
No
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
opsd_human |
|
MT1 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1A
|
MT1
|
Melatonin |
A (Rhodopsin) |
Human |
MT1 receptor |
6ME5 |
6me5 |
|
ETB receptor |
2022-06-19 |
Inactive |
Yes
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
5XPR |
5xpr |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
3UZC |
3uzc |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
7PX4 |
7px4 |
|
SST4 receptor |
2022-06-19 |
Active |
No
|
SSR4
|
SST4
|
Somatostatin |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
ssr4_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
7MTB |
7mtb |
|
ADGRB2 |
2022-06-19 |
Intermediate |
No
|
AGRB2
|
ADGRB2
|
ADGRB |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrb2_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
3D4S |
3d4s |
|
GPR132 |
2022-06-19 |
Intermediate |
No
|
GP132
|
GPR132
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gp132_human |
|
GAL2 receptor |
2022-06-19 |
Inactive |
No
|
GALR2
|
GAL2
|
Galanin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
galr2_human |
|
GAL2 receptor |
2022-06-19 |
Intermediate |
No
|
GALR2
|
GAL2
|
Galanin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
galr2_human |
|
GPR3 |
2022-06-19 |
Active |
No
|
GPR3
|
GPR3
|
A orphans |
A (Rhodopsin) |
Human |
S1P5 receptor |
7EW1 |
gpr3_human |
|
DP2 receptor |
2022-06-19 |
Inactive |
Yes
|
PD2R2
|
DP2
|
Prostanoid |
A (Rhodopsin) |
Human |
DP2 receptor |
7M8W |
7m8w |
|
BB2 receptor |
2022-06-19 |
Active |
No
|
GRPR
|
BB2
|
Bombesin |
A (Rhodopsin) |
Human |
GAL1 receptor |
7WQ3 |
grpr_human |
|
Rhodopsin |
2022-06-19 |
Inactive |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
1F88 |
1f88 |
|
CX3CR1 |
2022-06-19 |
Inactive |
No
|
CX3C1
|
CX3CR1
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
cx3c1_human |
|
GPR52 |
2022-06-19 |
Inactive |
Yes
|
GPR52
|
GPR52
|
A orphans |
A (Rhodopsin) |
Human |
GPR52 |
6LI0 |
6li0 |
|
β2-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
6MXT |
6mxt |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
7PYR |
7pyr |
|
UT receptor |
2022-06-19 |
Inactive |
No
|
UR2R
|
UT
|
Urotensin |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ur2r_human |
|
GPR132 |
2022-06-19 |
Active |
No
|
GP132
|
GPR132
|
A orphans |
A (Rhodopsin) |
Human |
AT2 receptor |
5UNG |
gp132_human |
|
GPR160 |
2022-06-19 |
Intermediate |
No
|
GP160
|
GPR160
|
A orphans |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4NTJ |
gp160_human |
|
MC2 receptor |
2022-06-19 |
Intermediate |
No
|
ACTHR
|
MC2
|
Melanocortin |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
acthr_human |
|
TAS2R42 |
2022-06-19 |
Intermediate |
No
|
T2R42
|
TAS2R42
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
t2r42_human |
|
5-HT1E receptor |
2022-06-19 |
Inactive |
No
|
5HT1E
|
5-HT1E
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAQ |
5ht1e_human |
|
GPR27 |
2022-06-19 |
Inactive |
No
|
GPR27
|
GPR27
|
A orphans |
A (Rhodopsin) |
Human |
D4 receptor |
5WIV |
gpr27_human |
|
PAR2 |
2022-06-19 |
Inactive |
No
|
PAR2
|
PAR2
|
Proteinase-activated |
A (Rhodopsin) |
Human |
CXCR4 |
3ODU |
par2_human |
|
GPR158 |
2022-06-19 |
Inactive |
Yes
|
GP158
|
GPR158
|
C Orphans |
C (Glutamate) |
Human |
GPR158 |
7EWR |
7ewr |
|
S1P5 receptor |
2022-06-19 |
Inactive |
No
|
S1PR5
|
S1P5
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
s1pr5_human |
|
P2RY8 |
2022-06-19 |
Active |
No
|
P2RY8
|
P2RY8
|
A orphans |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
p2ry8_human |
|
α2A-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADA2A
|
α2A
|
Adrenoceptors |
A (Rhodopsin) |
Human |
α2A-adrenoceptor |
6KUY |
6kuy |
|
GPR4 |
2022-06-19 |
Intermediate |
No
|
GPR4
|
GPR4
|
A orphans |
A (Rhodopsin) |
Human |
PAF receptor |
5ZKQ |
gpr4_human |
|
GPR22 |
2022-06-19 |
Inactive |
No
|
GPR22
|
GPR22
|
A orphans |
A (Rhodopsin) |
Human |
H1 receptor |
3RZE |
gpr22_human |
|
Rhodopsin |
2022-06-19 |
Inactive |
No
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
1U19 |
opsd_human |
|
TAS2R45 |
2022-06-19 |
Intermediate |
No
|
T2R45
|
TAS2R45
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2B receptor |
5TVN |
t2r45_human |
|
TAS2R42 |
2022-06-19 |
Active |
No
|
T2R42
|
TAS2R42
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
7DFL |
t2r42_human |
|
NK2 receptor |
2022-06-19 |
Active |
No
|
NK2R
|
NK2
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
7P00 |
nk2r_human |
|
GLP-1 receptor |
2022-06-19 |
Active |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
7LCK |
7lck |
|
CXCR4 |
2022-06-19 |
Active |
No
|
CXCR4
|
CXCR4
|
Chemokine |
A (Rhodopsin) |
Human |
CCR6 |
6WWZ |
cxcr4_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5VRA |
5vra |
|
M2 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M2 receptor |
5ZKB |
5zkb |
|
PAR1 |
2022-06-19 |
Inactive |
No
|
PAR1
|
PAR1
|
Proteinase-activated |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
par1_human |
|
D3 receptor |
2022-06-19 |
Inactive |
Yes
|
DRD3
|
D3
|
Dopamine |
A (Rhodopsin) |
Human |
D3 receptor |
3PBL |
3pbl |
|
LPA2 receptor |
2022-06-19 |
Active |
No
|
LPAR2
|
LPA2
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
LPA1 receptor |
7TD0 |
lpar2_human |
|
B1 receptor |
2022-06-19 |
Intermediate |
No
|
BKRB1
|
B1
|
Bradykinin |
A (Rhodopsin) |
Human |
GPR183 |
7TUY |
bkrb1_human |
|
DP2 receptor |
2022-06-19 |
Active |
No
|
PD2R2
|
DP2
|
Prostanoid |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
pd2r2_human |
|
NPFF1 receptor |
2022-06-19 |
Intermediate |
No
|
NPFF1
|
NPFF1
|
Neuropeptide FF/neuropeptide AF |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
npff1_human |
|
ADGRG5 |
2022-06-19 |
Intermediate |
No
|
AGRG5
|
ADGRG5
|
ADGRG |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrg5_human |
|
SST1 receptor |
2022-06-20 |
Inactive |
No
|
SSR1
|
SST1
|
Somatostatin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
ssr1_human |
|
CCR2 |
2022-06-19 |
Active |
No
|
CCR2
|
CCR2
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
7O7F |
ccr2_human |
|
GPR132 |
2022-06-19 |
Inactive |
No
|
GP132
|
GPR132
|
A orphans |
A (Rhodopsin) |
Human |
CCR7 |
6QZH |
gp132_human |
|
GHRH receptor |
2022-06-19 |
Inactive |
No
|
GHRHR
|
GHRH
|
Glucagon |
B1 (Secretin) |
Human |
PTH1 receptor |
6FJ3 |
ghrhr_human |
|
ACKR3 |
2022-06-19 |
Active |
No
|
ACKR3
|
ACKR3
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFO |
ackr3_human |
|
ADGRF5 |
2022-06-19 |
Inactive |
No
|
AGRF5
|
ADGRF5
|
ADGRF |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrf5_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TP6 |
6tp6 |
|
CCR1 |
2022-06-19 |
Inactive |
No
|
CCR1
|
CCR1
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ccr1_human |
|
kisspeptin receptor |
2022-06-19 |
Intermediate |
No
|
KISSR
|
kisspeptin
|
Kisspeptin |
A (Rhodopsin) |
Human |
PAR1 |
3VW7 |
kissr_human |
|
GPR37 |
2022-06-19 |
Active |
No
|
GPR37
|
GPR37
|
A orphans |
A (Rhodopsin) |
Human |
OX2 receptor |
7L1V |
gpr37_human |
|
μ receptor |
2022-06-19 |
Active |
No
|
OPRM
|
μ
|
Opioid |
A (Rhodopsin) |
Human |
μ receptor |
7U2L |
oprm_human |
|
ETB receptor |
2022-06-19 |
Inactive |
Yes
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
5X93 |
5x93 |
|
GPR153 |
2022-06-19 |
Intermediate |
No
|
GP153
|
GPR153
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp153_human |
|
MT1 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1A
|
MT1
|
Melatonin |
A (Rhodopsin) |
Human |
MT1 receptor |
6PS8 |
6ps8 |
|
MRGPRE |
2022-06-19 |
Active |
No
|
MRGRE
|
MRGPRE
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VDL |
mrgre_human |
|
ADGRF1 |
2022-06-19 |
Inactive |
No
|
AGRF1
|
ADGRF1
|
ADGRF |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrf1_human |
|
ADGRG2 |
2022-06-19 |
Inactive |
No
|
AGRG2
|
ADGRG2
|
ADGRG |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrg2_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5IU4 |
5iu4 |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5K2B |
5k2b |
|
GPR1 |
2022-06-19 |
Active |
No
|
GPR1
|
GPR1
|
A orphans |
A (Rhodopsin) |
Human |
FPR1 |
7WVU |
gpr1_human |
|
MC3 receptor |
2022-06-19 |
Active |
No
|
MC3R
|
MC3
|
Melanocortin |
A (Rhodopsin) |
Human |
MC4 receptor |
7F54 |
mc3r_human |
|
TAS2R42 |
2022-06-19 |
Inactive |
No
|
T2R42
|
TAS2R42
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
3RZE |
t2r42_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5OLH |
5olh |
|
Rhodopsin |
2022-06-19 |
Inactive |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
1GZM |
1gzm |
|
mGlu5 receptor |
2022-06-19 |
Active |
No
|
GRM5
|
mGlu5
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu4 receptor |
7E9H |
grm5_human |
|
CysLT1 receptor |
2022-06-19 |
Inactive |
No
|
CLTR1
|
CysLT1
|
Leukotriene |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
cltr1_human |
|
LGR5 |
2022-06-19 |
Intermediate |
No
|
LGR5
|
LGR5
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
lgr5_human |
|
GPR173 |
2022-06-19 |
Inactive |
No
|
GP173
|
GPR173
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2C receptor |
6BQH |
gp173_human |
|
κ receptor |
2022-06-19 |
Active |
Yes
|
OPRK
|
κ
|
Opioid |
A (Rhodopsin) |
Human |
κ receptor |
6B73 |
6b73 |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
4A4M |
4a4m |
|
FSH receptor |
2022-06-19 |
Inactive |
No
|
FSHR
|
FSH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
fshr_human |
|
GPR84 |
2022-06-19 |
Inactive |
No
|
GPR84
|
GPR84
|
A orphans |
A (Rhodopsin) |
Human |
ETB receptor |
5X93 |
gpr84_human |
|
NK2 receptor |
2022-06-19 |
Intermediate |
No
|
NK2R
|
NK2
|
Tachykinin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
nk2r_human |
|
TAS1R3 |
2022-06-20 |
Active |
No
|
TS1R3
|
TAS1R3
|
Taste 1 |
C (Glutamate) |
Human |
CaS receptor |
7DD6 |
ts1r3_human |
|
TAS2R8 |
2022-06-19 |
Intermediate |
No
|
TA2R8
|
TAS2R8
|
Taste 2 |
T (Taste 2) |
Human |
LPA6 receptor |
5XSZ |
ta2r8_human |
|
mGlu7 receptor |
2022-06-19 |
Intermediate |
No
|
GRM7
|
mGlu7
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
grm7_human |
|
GPR3 |
2022-06-19 |
Intermediate |
No
|
GPR3
|
GPR3
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
gpr3_human |
|
TSH receptor |
2022-06-19 |
Intermediate |
No
|
TSHR
|
TSH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
tshr_human |
|
GPRC5C |
2022-06-19 |
Inactive |
No
|
GPC5C
|
GPRC5C
|
C Orphans |
C (Glutamate) |
Human |
mGlu3 receptor |
7WIH |
gpc5c_human |
|
M3 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM3
|
M3
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Rat |
M3 receptor |
5ZHP |
5zhp |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5K2D |
5k2d |
|
AT1 receptor |
2022-06-19 |
Intermediate |
No
|
AGTR1
|
AT1
|
Angiotensin |
A (Rhodopsin) |
Human |
GPR183 |
7TUY |
agtr1_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
3PQR |
3pqr |
|
M2 receptor |
2022-06-19 |
Intermediate |
No
|
ACM2
|
M2
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
acm2_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5UIG |
5uig |
|
LGR4 |
2022-06-19 |
Active |
No
|
LGR4
|
LGR4
|
A orphans |
A (Rhodopsin) |
Human |
LH receptor |
7FIG |
lgr4_human |
|
GPR37L1 |
2022-06-19 |
Active |
No
|
G37L1
|
GPR37L1
|
A orphans |
A (Rhodopsin) |
Human |
MT1 receptor |
7VGZ |
g37l1_human |
|
CaS receptor |
2022-06-19 |
Active |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7SIM |
7sim |
|
A2A receptor |
2022-06-20 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5OLG |
5olg |
|
US28 |
2022-06-19 |
Active |
Yes
|
Q80KM9
|
US28
|
Unclassified |
A (Rhodopsin) |
strain AD169 |
US28 |
5WB2 |
5wb2 |
|
ETA receptor |
2022-06-19 |
Inactive |
No
|
EDNRA
|
ETA
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
5X93 |
ednra_human |
|
TAS2R4 |
2022-06-19 |
Intermediate |
No
|
TA2R4
|
TAS2R4
|
Taste 2 |
T (Taste 2) |
Human |
LPA6 receptor |
5XSZ |
ta2r4_human |
|
Y4 receptor |
2022-06-19 |
Active |
No
|
NPY4R
|
Y4
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
Y1 receptor |
7VGX |
npy4r_human |
|
ACKR2 |
2022-06-19 |
Active |
No
|
ACKR2
|
ACKR2
|
Chemokine |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
ackr2_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TP4 |
6tp4 |
|
5-HT2B receptor |
2022-06-19 |
Intermediate |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5tvn |
|
EP1 receptor |
2022-06-19 |
Intermediate |
No
|
PE2R1
|
EP1
|
Prostanoid |
A (Rhodopsin) |
Human |
TP receptor |
6IIV |
pe2r1_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5NLX |
5nlx |
|
GPR21 |
2022-06-19 |
Intermediate |
No
|
GPR21
|
GPR21
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr21_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
7ARO |
7aro |
|
MRGPRX2 |
2022-06-19 |
Active |
Yes
|
MRGX2
|
MRGPRX2
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VV6 |
7vv6 |
|
CysLT2 receptor |
2022-06-19 |
Active |
No
|
CLTR2
|
CysLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
cltr2_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TQ9 |
6tq9 |
|
MCH1 receptor |
2022-06-19 |
Inactive |
No
|
MCHR1
|
MCH1
|
Melanin-concentrating hormone |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
mchr1_human |
|
GPR45 |
2022-06-19 |
Active |
No
|
GPR45
|
GPR45
|
A orphans |
A (Rhodopsin) |
Human |
D2 receptor |
7JVR |
gpr45_human |
|
CysLT2 receptor |
2022-06-19 |
Intermediate |
Yes
|
CLTR2
|
CysLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
CysLT2 receptor |
6RZ7 |
6rz7 |
|
TAAR6 |
2022-06-19 |
Intermediate |
No
|
TAAR6
|
TAAR6
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
taar6_human |
|
M1 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM1
|
M1
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M1 receptor |
5CXV |
5cxv |
|
CXCR1 |
2022-06-19 |
Inactive |
No
|
CXCR1
|
CXCR1
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
cxcr1_human |
|
AT2 receptor |
2022-06-19 |
Active |
Yes
|
AGTR2
|
AT2
|
Angiotensin |
A (Rhodopsin) |
Human |
AT2 receptor |
5UNF |
5unf |
|
RXFP4 |
2022-06-19 |
Active |
No
|
RL3R2
|
RXFP4
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
AT1 receptor |
6DO1 |
rl3r2_human |
|
NTS1 receptor |
2022-06-19 |
Active |
Yes
|
NTR1
|
NTS1
|
Neurotensin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6PWC |
6pwc |
|
V1B receptor |
2022-06-19 |
Intermediate |
No
|
V1BR
|
V1B
|
Vasopressin and oxytocin |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
v1br_human |
|
XCR1 |
2022-06-19 |
Inactive |
No
|
XCR1
|
XCR1
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
xcr1_human |
|
κ receptor |
2022-06-19 |
Inactive |
Yes
|
OPRK
|
κ
|
Opioid |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
4djh |
|
H4 receptor |
2022-06-19 |
Inactive |
No
|
HRH4
|
H4
|
Histamine |
A (Rhodopsin) |
Human |
M3 receptor |
5ZHP |
hrh4_human |
|
A2A receptor |
2022-06-19 |
Intermediate |
No
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
aa2ar_human |
|
ADGRE1 |
2022-06-19 |
Inactive |
No
|
AGRE1
|
ADGRE1
|
ADGRE |
B2 (Adhesion) |
Human |
calcitonin receptor-like receptor |
7KNU |
agre1_human |
|
GLP-1 receptor |
2022-06-19 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
6KK1 |
6kk1 |
|
GPR88 |
2022-06-19 |
Inactive |
No
|
GPR88
|
GPR88
|
A orphans |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
gpr88_human |
|
Y1 receptor |
2022-06-19 |
Intermediate |
No
|
NPY1R
|
Y1
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
npy1r_human |
|
calcitonin receptor-like receptor |
2022-06-19 |
Intermediate |
No
|
CALRL
|
calcitonin-like
|
Calcitonin |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
calrl_human |
|
GPR27 |
2022-06-19 |
Active |
No
|
GPR27
|
GPR27
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2C receptor |
6BQG |
gpr27_human |
|
GPR17 |
2022-06-19 |
Inactive |
No
|
GPR17
|
GPR17
|
A orphans |
A (Rhodopsin) |
Human |
apelin receptor |
5VBL |
gpr17_human |
|
5-HT4 receptor |
2022-06-19 |
Active |
No
|
5HT4R
|
5-HT4
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
D1 receptor |
7JVQ |
5ht4r_human |
|
TAS2R39 |
2022-06-19 |
Active |
No
|
T2R39
|
TAS2R39
|
Taste 2 |
T (Taste 2) |
Human |
κ receptor |
6B73 |
t2r39_human |
|
GPBA receptor |
2022-06-19 |
Inactive |
No
|
GPBAR
|
GPBA
|
Bile acid |
A (Rhodopsin) |
Human |
CB1 receptor |
5TGZ |
gpbar_human |
|
Rhodopsin |
2022-06-19 |
Inactive |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
3C9L |
3c9l |
|
ADGRF3 |
2022-06-19 |
Intermediate |
No
|
AGRF3
|
ADGRF3
|
ADGRF |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrf3_human |
|
GPR119 |
2022-06-19 |
Intermediate |
No
|
GP119
|
GPR119
|
GPR18, GPR55 and GPR119 |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp119_human |
|
GnRH1 receptor |
2022-06-19 |
Active |
No
|
GNRHR
|
GnRH1
|
Gonadotrophin-releasing hormone |
A (Rhodopsin) |
Human |
OT receptor |
7RYC |
gnrhr_human |
|
FPR3 |
2022-06-19 |
Inactive |
No
|
FPR3
|
FPR3
|
Formylpeptide |
A (Rhodopsin) |
Human |
DP2 receptor |
7M8W |
fpr3_human |
|
AT1 receptor |
2022-06-19 |
Inactive |
Yes
|
AGTR1
|
AT1
|
Angiotensin |
A (Rhodopsin) |
Human |
AT1 receptor |
4YAY |
4yay |
|
Y2 receptor |
2022-06-19 |
Inactive |
Yes
|
NPY2R
|
Y2
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
Y2 receptor |
7DDZ |
7ddz |
|
mGlu4 receptor |
2022-06-19 |
Inactive |
No
|
GRM4
|
mGlu4
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu7 receptor |
7EPC |
grm4_human |
|
H2 receptor |
2022-06-19 |
Active |
No
|
HRH2
|
H2
|
Histamine |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BU7 |
hrh2_human |
|
MRGPRX3 |
2022-06-19 |
Active |
No
|
MRGX3
|
MRGPRX3
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX4 |
7S8P |
mrgx3_human |
|
FFA4 receptor |
2022-06-19 |
Active |
No
|
FFAR4
|
FFA4
|
Free fatty acid |
A (Rhodopsin) |
Human |
CCK2 receptor |
7F8W |
ffar4_human |
|
ACKR1 |
2022-06-19 |
Intermediate |
No
|
ACKR1
|
ACKR1
|
Chemokine |
A (Rhodopsin) |
Human |
P2Y1 receptor |
4XNW |
ackr1_human |
|
S1P3 receptor |
2022-06-19 |
Active |
Yes
|
S1PR3
|
S1P3
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P3 receptor |
7C4S |
7c4s |
|
GPR142 |
2022-06-19 |
Active |
No
|
GP142
|
GPR142
|
A orphans |
A (Rhodopsin) |
Human |
GPR139 |
7VUG |
gp142_human |
|
GPR37L1 |
2022-06-19 |
Intermediate |
No
|
G37L1
|
GPR37L1
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
g37l1_human |
|
P2Y11 receptor |
2022-06-19 |
Intermediate |
No
|
P2Y11
|
P2Y11
|
P2Y |
A (Rhodopsin) |
Human |
P2Y1 receptor |
4XNW |
p2y11_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
5F8U |
5f8u |
|
CCK2 receptor |
2022-06-19 |
Intermediate |
No
|
GASR
|
CCK2
|
Cholecystokinin |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gasr_human |
|
kisspeptin receptor |
2022-06-19 |
Active |
No
|
KISSR
|
kisspeptin
|
Kisspeptin |
A (Rhodopsin) |
Human |
GAL1 receptor |
7WQ3 |
kissr_human |
|
P2Y12 receptor |
2022-06-19 |
Intermediate |
Yes
|
P2Y12
|
P2Y12
|
P2Y |
A (Rhodopsin) |
Human |
P2Y12 receptor |
4PXZ |
4pxz |
|
LH receptor |
2022-06-19 |
Inactive |
Yes
|
LSHR
|
LH
|
Glycoprotein hormone |
A (Rhodopsin) |
Human |
LH receptor |
7FIJ |
7fij |
|
CRF1 receptor |
2022-06-19 |
Intermediate |
No
|
CRFR1
|
CRF1
|
Corticotropin-releasing factor |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
crfr1_human |
|
CXCR3 |
2022-06-19 |
Active |
No
|
CXCR3
|
CXCR3
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFO |
cxcr3_human |
|
ADGRA1 |
2022-06-19 |
Inactive |
No
|
AGRA1
|
ADGRA1
|
ADGRA |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agra1_human |
|
ADGRF2 |
2022-06-19 |
Inactive |
No
|
AGRF2
|
ADGRF2
|
ADGRF |
B2 (Adhesion) |
Human |
calcitonin receptor-like receptor |
7KNU |
agrf2_human |
|
GPR32 |
2022-06-19 |
Intermediate |
No
|
GPR32
|
GPR32
|
A orphans |
A (Rhodopsin) |
Human |
P2Y1 receptor |
4XNW |
gpr32_human |
|
GPR27 |
2022-06-19 |
Intermediate |
No
|
GPR27
|
GPR27
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr27_human |
|
PTH1 receptor |
2021-11-02 |
Inactive |
Yes
|
PTH1R
|
PTH1
|
Parathyroid hormone |
B1 (Secretin) |
Human |
PTH1 receptor |
6FJ3 |
6fj3 |
|
mGlu2 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM2
|
mGlu2
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu2 receptor |
7EPA |
7epa |
|
MRGPRX2 |
2022-06-19 |
Intermediate |
No
|
MRGX2
|
MRGPRX2
|
A orphans |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
mrgx2_human |
|
S1P3 receptor |
2022-06-19 |
Inactive |
No
|
S1PR3
|
S1P3
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
s1pr3_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5NM2 |
5nm2 |
|
EP3 receptor |
2022-06-19 |
Intermediate |
No
|
PE2R3
|
EP3
|
Prostanoid |
A (Rhodopsin) |
Human |
TP receptor |
6IIV |
pe2r3_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5OLV |
5olv |
|
GPR101 |
2022-06-19 |
Inactive |
No
|
GP101
|
GPR101
|
A orphans |
A (Rhodopsin) |
Human |
α1B-adrenoceptor |
7B6W |
gp101_human |
|
β1-adrenoceptor |
2022-06-20 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
2YCW |
2ycw |
|
BB2 receptor |
2022-06-19 |
Intermediate |
No
|
GRPR
|
BB2
|
Bombesin |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
grpr_human |
|
S1P2 receptor |
2022-06-19 |
Inactive |
No
|
S1PR2
|
S1P2
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
s1pr2_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
7WC5 |
7wc5 |
|
CaS receptor |
2022-06-19 |
Active |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7M3G |
7m3g |
|
ADGRB3 |
2022-06-19 |
Intermediate |
No
|
AGRB3
|
ADGRB3
|
ADGRB |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrb3_human |
|
ADGRG1 |
2022-06-19 |
Inactive |
No
|
AGRG1
|
ADGRG1
|
ADGRG |
B2 (Adhesion) |
Human |
glucagon receptor |
5YQZ |
agrg1_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6LPL |
6lpl |
|
β2-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
6E67 |
6e67 |
|
SMO |
2022-06-20 |
Inactive |
Yes
|
SMO
|
SMO
|
Frizzled |
F (Frizzled) |
Human |
SMO |
4QIM |
4qim |
|
M4 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM4
|
M4
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M4 receptor |
5DSG |
5dsg |
|
MC5 receptor |
2022-06-19 |
Intermediate |
No
|
MC5R
|
MC5
|
Melanocortin |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
mc5r_human |
|
TAS2R38 |
2022-06-19 |
Active |
No
|
T2R38
|
TAS2R38
|
Taste 2 |
T (Taste 2) |
Human |
AT1 receptor |
6DO1 |
t2r38_human |
|
C5a2 receptor |
2022-06-19 |
Intermediate |
No
|
C5AR2
|
C5a2
|
Complement peptide |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
c5ar2_human |
|
ADGRG4 |
2022-06-19 |
Inactive |
No
|
AGRG4
|
ADGRG4
|
ADGRG |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrg4_human |
|
TAS1R2 |
2022-06-19 |
Intermediate |
No
|
TS1R2
|
TAS1R2
|
Taste 1 |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
ts1r2_human |
|
B1 receptor |
2022-06-19 |
Inactive |
No
|
BKRB1
|
B1
|
Bradykinin |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
bkrb1_human |
|
GPR75 |
2022-06-19 |
Intermediate |
No
|
GPR75
|
GPR75
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr75_human |
|
MRGPRF |
2022-06-19 |
Active |
No
|
MRGRF
|
MRGPRF
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX2 |
7VDL |
mrgrf_human |
|
TAAR5 |
2022-06-19 |
Active |
No
|
TAAR5
|
TAAR5
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1B receptor |
6G79 |
taar5_human |
|
AT1 receptor |
2022-06-20 |
Active |
Yes
|
AGTR1
|
AT1
|
Angiotensin |
A (Rhodopsin) |
Human |
AT1 receptor |
6OS1 |
6os1 |
|
GPR18 |
2022-06-19 |
Inactive |
No
|
GPR18
|
GPR18
|
GPR18, GPR55 and GPR119 |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
gpr18_human |
|
β2-adrenoceptor |
2022-06-20 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
3NY9 |
3ny9 |
|
GPR139 |
2022-06-19 |
Intermediate |
No
|
GP139
|
GPR139
|
A orphans |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
gp139_human |
|
MCH2 receptor |
2022-06-19 |
Active |
No
|
MCHR2
|
MCH2
|
Melanin-concentrating hormone |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
mchr2_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6PS7 |
6ps7 |
|
β2-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
adrb2_human |
|
mGlu2 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM2
|
mGlu2
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu2 receptor |
7EPF |
7epf |
|
GPRC6 receptor |
2022-06-19 |
Inactive |
No
|
GPC6A
|
GPRC6
|
C Orphans |
C (Glutamate) |
Human |
CaS receptor |
7DD5 |
gpc6a_human |
|
β1-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
6H7L |
6h7l |
|
Rhodopsin |
2022-06-20 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6FKD |
6fkd |
|
GPR68 |
2022-06-19 |
Active |
No
|
OGR1
|
GPR68
|
A orphans |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
ogr1_human |
|
ADGRE2 |
2022-06-19 |
Inactive |
No
|
AGRE2
|
ADGRE2
|
ADGRE |
B2 (Adhesion) |
Human |
GLP-1 receptor |
6LN2 |
agre2_human |
|
NTS1 receptor |
2022-06-19 |
Active |
Yes
|
NTR1
|
NTS1
|
Neurotensin |
A (Rhodopsin) |
Rat |
NTS1 receptor |
4XES |
4xes |
|
TAS2R4 |
2022-06-19 |
Active |
No
|
TA2R4
|
TAS2R4
|
Taste 2 |
T (Taste 2) |
Human |
5-HT1B receptor |
6G79 |
ta2r4_human |
|
secretin receptor |
2022-06-19 |
Intermediate |
No
|
SCTR
|
secretin
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
sctr_human |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
5D5B |
5d5b |
|
MT2 receptor |
2022-06-19 |
Inactive |
Yes
|
MTR1B
|
MT2
|
Melatonin |
A (Rhodopsin) |
Human |
MT2 receptor |
6ME6 |
6me6 |
|
β2-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
3P0G |
3p0g |
|
GPR62 |
2022-06-19 |
Active |
No
|
GPR62
|
GPR62
|
A orphans |
A (Rhodopsin) |
Human |
D3 receptor |
7CMV |
gpr62_human |
|
B2 receptor |
2022-06-19 |
Inactive |
No
|
BKRB2
|
B2
|
Bradykinin |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
bkrb2_human |
|
EP3 receptor |
2022-06-19 |
Inactive |
No
|
PE2R3
|
EP3
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
pe2r3_human |
|
BB1 receptor |
2022-06-19 |
Inactive |
No
|
NMBR
|
BB1
|
Bombesin |
A (Rhodopsin) |
Human |
ETB receptor |
5X93 |
nmbr_human |
|
FZD5 |
2022-06-19 |
Inactive |
Yes
|
FZD5
|
FZD5
|
Frizzled |
F (Frizzled) |
Human |
FZD5 |
6WW2 |
6ww2 |
|
FFA1 receptor |
2022-06-19 |
Intermediate |
Yes
|
FFAR1
|
FFA1
|
Free fatty acid |
A (Rhodopsin) |
Human |
FFA1 receptor |
5TZR |
5tzr |
|
CB1 receptor |
2022-06-19 |
Active |
Yes
|
CNR1
|
CB1
|
Cannabinoid |
A (Rhodopsin) |
Human |
CB1 receptor |
7V3Z |
7v3z |
|
GPR35 |
2022-06-19 |
Inactive |
No
|
GPR35
|
GPR35
|
A orphans |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
gpr35_human |
|
P2Y1 receptor |
2022-06-19 |
Active |
No
|
P2RY1
|
P2Y1
|
P2Y |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
p2ry1_human |
|
GABAB2 |
2022-06-19 |
Active |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
6UO8 |
6uo8 |
|
FZD2 |
2022-06-19 |
Active |
No
|
FZD2
|
FZD2
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd2_human |
|
mGlu2 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM2
|
mGlu2
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu2 receptor |
7EPE |
7epe |
|
ADGRF4 |
2022-06-19 |
Intermediate |
No
|
AGRF4
|
ADGRF4
|
ADGRF |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrf4_human |
|
NPBW2 receptor |
2022-06-19 |
Inactive |
No
|
NPBW2
|
NPBW2
|
Neuropeptide W/neuropeptide B |
A (Rhodopsin) |
Human |
δ receptor |
4N6H |
npbw2_human |
|
GPR34 |
2022-06-19 |
Inactive |
No
|
GPR34
|
GPR34
|
A orphans |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
gpr34_human |
|
GPR158 |
2022-06-19 |
Inactive |
Yes
|
GP158
|
GPR158
|
C Orphans |
C (Glutamate) |
Human |
GPR158 |
7SHE |
7she |
|
S1P1 receptor |
2022-06-19 |
Inactive |
Yes
|
S1PR1
|
S1P1
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
3v2y |
|
ETA receptor |
2022-06-19 |
Intermediate |
No
|
EDNRA
|
ETA
|
Endothelin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
ednra_human |
|
MT1 receptor |
2022-06-19 |
Intermediate |
No
|
MTR1A
|
MT1
|
Melatonin |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
mtr1a_human |
|
HCA1 receptor |
2022-06-19 |
Active |
No
|
HCAR1
|
HCA1
|
Hydroxycarboxylic acid |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
hcar1_human |
|
succinate receptor |
2022-06-19 |
Active |
No
|
SUCR1
|
succinate
|
Succinate |
A (Rhodopsin) |
Human |
GAL1 receptor |
7WQ3 |
sucr1_human |
|
GLP-1 receptor |
2022-06-19 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
6KK7 |
6kk7 |
|
GPR25 |
2022-06-19 |
Active |
No
|
GPR25
|
GPR25
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
6DO1 |
gpr25_human |
|
ADGRE5 |
2022-06-19 |
Active |
No
|
AGRE5
|
ADGRE5
|
ADGRE |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agre5_human |
|
PAR2 |
2022-06-19 |
Active |
No
|
PAR2
|
PAR2
|
Proteinase-activated |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
par2_human |
|
GPR148 |
2022-06-19 |
Active |
No
|
GP148
|
GPR148
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1D receptor |
7E32 |
gp148_human |
|
ADGRB2 |
2022-06-19 |
Active |
No
|
AGRB2
|
ADGRB2
|
ADGRB |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agrb2_human |
|
CCK1 receptor |
2022-06-19 |
Inactive |
Yes
|
CCKAR
|
CCK1
|
Cholecystokinin |
A (Rhodopsin) |
Human |
CCK1 receptor |
7F8Y |
7f8y |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
4AMI |
4ami |
|
PKR1 |
2022-06-19 |
Inactive |
No
|
PKR1
|
PKR1
|
Prokineticin |
A (Rhodopsin) |
Human |
Y2 receptor |
7DDZ |
pkr1_human |
|
A2B receptor |
2022-06-19 |
Intermediate |
No
|
AA2BR
|
A2B
|
Adenosine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
aa2br_human |
|
ETB receptor |
2022-06-19 |
Inactive |
Yes
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ETB receptor |
6LRY |
6lry |
|
FFA1 receptor |
2022-06-19 |
Inactive |
No
|
FFAR1
|
FFA1
|
Free fatty acid |
A (Rhodopsin) |
Human |
CCK1 receptor |
7F8Y |
ffar1_human |
|
oxoglutarate receptor |
2022-06-19 |
Active |
No
|
OXGR1
|
oxoglutarate
|
Oxoglutarate |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
oxgr1_human |
|
FZD2 |
2022-06-19 |
Inactive |
No
|
FZD2
|
FZD2
|
Frizzled |
F (Frizzled) |
Human |
FZD5 |
6WW2 |
fzd2_human |
|
GLP-1 receptor |
2022-06-19 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5VEX |
5vex |
|
TAS2R13 |
2022-06-19 |
Inactive |
No
|
T2R13
|
TAS2R13
|
Taste 2 |
T (Taste 2) |
Human |
apelin receptor |
5VBL |
t2r13_human |
|
ghrelin receptor |
2022-06-19 |
Inactive |
Yes
|
GHSR
|
ghrelin
|
Ghrelin |
A (Rhodopsin) |
Human |
ghrelin receptor |
7F83 |
7f83 |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
4AMJ |
4amj |
|
GPR156 |
2022-06-19 |
Inactive |
No
|
GP156
|
GPR156
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
6WIV |
gp156_human |
|
GPR142 |
2022-06-19 |
Intermediate |
No
|
GP142
|
GPR142
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp142_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
5MZJ |
5mzj |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
3ZPR |
3zpr |
|
HCA2 receptor |
2022-06-19 |
Active |
No
|
HCAR2
|
HCA2
|
Hydroxycarboxylic acid |
A (Rhodopsin) |
Human |
κ receptor |
6B73 |
hcar2_human |
|
S1P1 receptor |
2022-06-19 |
Intermediate |
No
|
S1PR1
|
S1P1
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
s1pr1_human |
|
OPN1MW |
2022-06-19 |
Active |
No
|
OPSG
|
OPN1MW
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
4X1H |
opsg_human |
|
ACKR2 |
2022-06-19 |
Inactive |
No
|
ACKR2
|
ACKR2
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ackr2_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
7bvq |
|
PAF receptor |
2022-06-19 |
Active |
No
|
PTAFR
|
PAF
|
Platelet-activating factor |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
ptafr_human |
|
OX1 receptor |
2022-06-19 |
Inactive |
Yes
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
OX1 receptor |
6TOT |
6tot |
|
GPR101 |
2022-06-19 |
Intermediate |
No
|
GP101
|
GPR101
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp101_human |
|
GPR149 |
2022-06-19 |
Inactive |
No
|
GP149
|
GPR149
|
A orphans |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
gp149_human |
|
GABAB2 |
2022-06-19 |
Inactive |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
7CUM |
7cum |
|
Olfactory receptor 1A1 |
2022-06-19 |
Intermediate |
No
|
OR1A1
|
Olfactory 1A1
|
Olfactory |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
or1a1_human |
|
GABAB2 |
2022-06-19 |
Inactive |
Yes
|
GABR2
|
GABAB2
|
GABAB |
C (Glutamate) |
Human |
GABAB2 |
6UO9 |
6uo9 |
|
PTH2 receptor |
2022-06-19 |
Inactive |
No
|
PTH2R
|
PTH2
|
Parathyroid hormone |
B1 (Secretin) |
Human |
PTH1 receptor |
6FJ3 |
pth2r_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6AQF |
6aqf |
|
OT receptor |
2022-06-19 |
Intermediate |
No
|
OXYR
|
OT
|
Vasopressin and oxytocin |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
oxyr_human |
|
GPR141 |
2022-06-19 |
Intermediate |
No
|
GP141
|
GPR141
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gp141_human |
|
H2 receptor |
2022-06-19 |
Intermediate |
No
|
HRH2
|
H2
|
Histamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
hrh2_human |
|
TAS2R9 |
2022-06-19 |
Intermediate |
No
|
TA2R9
|
TAS2R9
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2B receptor |
5TVN |
ta2r9_human |
|
TAS2R43 |
2022-06-19 |
Intermediate |
No
|
T2R43
|
TAS2R43
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
t2r43_human |
|
BLT1 receptor |
2022-06-19 |
Intermediate |
No
|
LT4R1
|
BLT1
|
Leukotriene |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
lt4r1_human |
|
NTS2 receptor |
2022-06-19 |
Active |
No
|
NTR2
|
NTS2
|
Neurotensin |
A (Rhodopsin) |
Human |
NTS1 receptor |
4XES |
ntr2_human |
|
TAS2R40 |
2022-06-19 |
Intermediate |
No
|
T2R40
|
TAS2R40
|
Taste 2 |
T (Taste 2) |
Human |
LPA6 receptor |
5XSZ |
t2r40_human |
|
5-HT5A receptor |
2022-06-19 |
Active |
No
|
5HT5A
|
5-HT5A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1D receptor |
7E32 |
5ht5a_human |
|
LGR6 |
2022-06-19 |
Intermediate |
No
|
LGR6
|
LGR6
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
lgr6_human |
|
succinate receptor |
2022-06-19 |
Intermediate |
No
|
SUCR1
|
succinate
|
Succinate |
A (Rhodopsin) |
Human |
succinate receptor |
6RNK |
sucr1_human |
|
OXE receptor |
2022-06-19 |
Inactive |
No
|
OXER1
|
OXE
|
Leukotriene |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
oxer1_human |
|
Y1 receptor |
2022-06-19 |
Inactive |
Yes
|
NPY1R
|
Y1
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
Y1 receptor |
5ZBH |
5zbh |
|
GPR135 |
2022-06-19 |
Intermediate |
No
|
GP135
|
GPR135
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gp135_human |
|
PAR2 |
2022-06-19 |
Intermediate |
Yes
|
PAR2
|
PAR2
|
Proteinase-activated |
A (Rhodopsin) |
Human |
PAR2 |
5NJ6 |
5nj6 |
|
CCR5 |
2021-11-02 |
Inactive |
Yes
|
CCR5
|
CCR5
|
Chemokine |
A (Rhodopsin) |
Human |
CCR5 |
7F1T |
7f1t |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
3RFM |
3rfm |
|
Rhodopsin |
2022-06-19 |
Inactive |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Japanese flying squid |
Rhodopsin |
2Z73 |
2z73 |
|
TAS2R30 |
2022-06-19 |
Active |
No
|
T2R30
|
TAS2R30
|
Taste 2 |
T (Taste 2) |
Human |
5-HT2C receptor |
6BQG |
t2r30_human |
|
SST5 receptor |
2022-06-19 |
Active |
No
|
SSR5
|
SST5
|
Somatostatin |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
ssr5_human |
|
IP receptor |
2022-06-19 |
Intermediate |
No
|
PI2R
|
IP
|
Prostanoid |
A (Rhodopsin) |
Human |
TP receptor |
6IIV |
pi2r_human |
|
GLP-2 receptor |
2022-06-19 |
Intermediate |
No
|
GLP2R
|
GLP-2
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
glp2r_human |
|
Y4 receptor |
2022-06-19 |
Inactive |
No
|
NPY4R
|
Y4
|
Neuropeptide Y |
A (Rhodopsin) |
Human |
Y1 receptor |
5ZBH |
npy4r_human |
|
EP4 receptor |
2022-06-19 |
Inactive |
Yes
|
PE2R4
|
EP4
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
5ywy |
|
D4 receptor |
2022-06-19 |
Inactive |
Yes
|
DRD4
|
D4
|
Dopamine |
A (Rhodopsin) |
Mouse |
D4 receptor |
6IQL |
6iql |
|
QRFP receptor |
2022-06-19 |
Inactive |
No
|
QRFPR
|
QRFP
|
Peptide P518 |
A (Rhodopsin) |
Human |
OX2 receptor |
5WQC |
qrfpr_human |
|
OX1 receptor |
2022-06-19 |
Intermediate |
No
|
OX1R
|
OX1
|
Orexin |
A (Rhodopsin) |
Human |
NTS1 receptor |
6Z8N |
ox1r_human |
|
5-HT1D receptor |
2022-06-19 |
Inactive |
No
|
5HT1D
|
5-HT1D
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAQ |
5ht1d_human |
|
GPR37 |
2022-06-19 |
Inactive |
No
|
GPR37
|
GPR37
|
A orphans |
A (Rhodopsin) |
Human |
ETB receptor |
5X93 |
gpr37_human |
|
β1-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
adrb1_human |
|
VPAC1 receptor |
2022-06-19 |
Inactive |
No
|
VIPR1
|
VPAC1
|
VIP and PACAP |
B1 (Secretin) |
Human |
PTH1 receptor |
6FJ3 |
vipr1_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6WGT |
6wgt |
|
BLT2 receptor |
2022-06-19 |
Intermediate |
No
|
LT4R2
|
BLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
lt4r2_human |
|
TAS2R60 |
2022-06-19 |
Intermediate |
No
|
T2R60
|
TAS2R60
|
Taste 2 |
T (Taste 2) |
Human |
PAR1 |
3VW7 |
t2r60_human |
|
OPN4 |
2022-06-19 |
Active |
No
|
OPN4
|
OPN4
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
4X1H |
opn4_human |
|
GHRH receptor |
2022-06-19 |
Intermediate |
No
|
GHRHR
|
GHRH
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
ghrhr_human |
|
CysLT1 receptor |
2022-06-19 |
Active |
No
|
CLTR1
|
CysLT1
|
Leukotriene |
A (Rhodopsin) |
Human |
AT1 receptor |
6DO1 |
cltr1_human |
|
NTS1 receptor |
2022-06-19 |
Active |
Yes
|
NTR1
|
NTS1
|
Neurotensin |
A (Rhodopsin) |
Rat |
NTS1 receptor |
4XEE |
4xee |
|
MRGPRX1 |
2022-06-19 |
Active |
No
|
MRGX1
|
MRGPRX1
|
A orphans |
A (Rhodopsin) |
Human |
MRGPRX4 |
7S8P |
mrgx1_human |
|
mGlu8 receptor |
2022-06-19 |
Active |
No
|
GRM8
|
mGlu8
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu4 receptor |
7E9H |
grm8_human |
|
ADGRG3 |
2022-06-19 |
Intermediate |
No
|
AGRG3
|
ADGRG3
|
ADGRG |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrg3_human |
|
GLP-1 receptor |
2022-06-20 |
Inactive |
Yes
|
GLP1R
|
GLP-1
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5VEW |
5vew |
|
PKR2 |
2022-06-19 |
Active |
No
|
PKR2
|
PKR2
|
Prokineticin |
A (Rhodopsin) |
Human |
NK1 receptor |
7P00 |
pkr2_human |
|
TAS2R16 |
2022-06-19 |
Inactive |
No
|
T2R16
|
TAS2R16
|
Taste 2 |
T (Taste 2) |
Human |
DP2 receptor |
7M8W |
t2r16_human |
|
D4 receptor |
2022-06-19 |
Inactive |
Yes
|
DRD4
|
D4
|
Dopamine |
A (Rhodopsin) |
Human |
D4 receptor |
5WIU |
5wiu |
|
GPR179 |
2022-06-19 |
Intermediate |
No
|
GP179
|
GPR179
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
7CA5 |
gp179_human |
|
M3 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM3
|
M3
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Rat |
M3 receptor |
4U16 |
4u16 |
|
β3-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADRB3
|
β3
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
adrb3_human |
|
CysLT2 receptor |
2022-06-19 |
Inactive |
No
|
CLTR2
|
CysLT2
|
Leukotriene |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
cltr2_human |
|
A3 receptor |
2022-06-19 |
Active |
No
|
AA3R
|
A3
|
Adenosine |
A (Rhodopsin) |
Human |
A1 receptor |
6D9H |
aa3r_human |
|
β1-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
6TKO |
6tko |
|
mGlu1 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM1
|
mGlu1
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu1 receptor |
4OR2 |
4or2 |
|
GPR160 |
2022-06-19 |
Active |
No
|
GP160
|
GPR160
|
A orphans |
A (Rhodopsin) |
Human |
H1 receptor |
7DFL |
gp160_human |
|
OPN1LW |
2022-06-19 |
Inactive |
No
|
OPSR
|
OPN1LW
|
Opsins |
A (Rhodopsin) |
Human |
Rhodopsin |
1U19 |
opsr_human |
|
ADGRL1 |
2022-06-19 |
Intermediate |
No
|
AGRL1
|
ADGRL1
|
ADGRL |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agrl1_human |
|
NPFF2 receptor |
2022-06-19 |
Active |
No
|
NPFF2
|
NPFF2
|
Neuropeptide FF/neuropeptide AF |
A (Rhodopsin) |
Human |
OX2 receptor |
7L1V |
npff2_human |
|
TAAR9 |
2022-06-19 |
Inactive |
No
|
TAAR9
|
TAAR9
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAQ |
taar9_human |
|
GPR1 |
2022-06-19 |
Inactive |
No
|
GPR1
|
GPR1
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
gpr1_human |
|
PKR1 |
2022-06-19 |
Active |
No
|
PKR1
|
PKR1
|
Prokineticin |
A (Rhodopsin) |
Human |
NK1 receptor |
7P00 |
pkr1_human |
|
FFA3 receptor |
2022-06-19 |
Active |
No
|
FFAR3
|
FFA3
|
Free fatty acid |
A (Rhodopsin) |
Human |
GPR183 |
7TUZ |
ffar3_human |
|
FZD9 |
2022-06-19 |
Active |
No
|
FZD9
|
FZD9
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd9_human |
|
α1A-adrenoceptor |
2022-06-19 |
Intermediate |
No
|
ADA1A
|
α1A
|
Adrenoceptors |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
ada1a_human |
|
CXCR6 |
2022-06-19 |
Active |
No
|
CXCR6
|
CXCR6
|
Chemokine |
A (Rhodopsin) |
Human |
CCR6 |
6WWZ |
cxcr6_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
2Y04 |
2y04 |
|
ADGRE3 |
2022-06-19 |
Inactive |
No
|
AGRE3
|
ADGRE3
|
ADGRE |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agre3_human |
|
ACKR1 |
2022-06-19 |
Active |
No
|
ACKR1
|
ACKR1
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFO |
ackr1_human |
|
AT2 receptor |
2022-06-19 |
Active |
Yes
|
AGTR2
|
AT2
|
Angiotensin |
A (Rhodopsin) |
Human |
AT2 receptor |
5UNG |
5ung |
|
PAR4 |
2022-06-19 |
Active |
No
|
PAR4
|
PAR4
|
Proteinase-activated |
A (Rhodopsin) |
Human |
FPR2/ALX |
7WVX |
par4_human |
|
μ receptor |
2022-06-19 |
Intermediate |
No
|
OPRM
|
μ
|
Opioid |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
oprm_human |
|
5-HT1B receptor |
2022-06-19 |
Intermediate |
No
|
5HT1B
|
5-HT1B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht1b_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6NWE |
6nwe |
|
BB1 receptor |
2022-06-19 |
Intermediate |
No
|
NMBR
|
BB1
|
Bombesin |
A (Rhodopsin) |
Human |
succinate receptor |
6RNK |
nmbr_human |
|
TAS2R14 |
2022-06-19 |
Active |
No
|
T2R14
|
TAS2R14
|
Taste 2 |
T (Taste 2) |
Human |
D2 receptor |
7JVR |
t2r14_human |
|
GLP-2 receptor |
2022-06-19 |
Inactive |
No
|
GLP2R
|
GLP-2
|
Glucagon |
B1 (Secretin) |
Human |
glucagon receptor |
5YQZ |
glp2r_human |
|
RXFP3 |
2022-06-19 |
Active |
No
|
RL3R1
|
RXFP3
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
rl3r1_human |
|
MRGPRX3 |
2022-06-19 |
Intermediate |
No
|
MRGX3
|
MRGPRX3
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
mrgx3_human |
|
β1-adrenoceptor |
2022-06-19 |
Active |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BU7 |
7bu7 |
|
GPR68 |
2022-06-19 |
Inactive |
No
|
OGR1
|
GPR68
|
A orphans |
A (Rhodopsin) |
Human |
CCR5 |
4MBS |
ogr1_human |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6FK7 |
6fk7 |
|
5-HT2B receptor |
2022-06-19 |
Active |
Yes
|
5HT2B
|
5-HT2B
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TUD |
5tud |
|
PAF receptor |
2022-06-19 |
Intermediate |
Yes
|
PTAFR
|
PAF
|
Platelet-activating factor |
A (Rhodopsin) |
Human |
PAF receptor |
5ZKQ |
5zkq |
|
S1P4 receptor |
2022-06-19 |
Intermediate |
No
|
S1PR4
|
S1P4
|
Lysophospholipid (S1P) |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
s1pr4_human |
|
P2Y14 receptor |
2022-06-19 |
Inactive |
No
|
P2Y14
|
P2Y14
|
P2Y |
A (Rhodopsin) |
Human |
CCR2 |
5T1A |
p2y14_human |
|
TAAR6 |
2022-06-19 |
Inactive |
No
|
TAAR6
|
TAAR6
|
A orphans |
A (Rhodopsin) |
Human |
5-HT1B receptor |
4IAQ |
taar6_human |
|
mGlu7 receptor |
2022-06-19 |
Active |
No
|
GRM7
|
mGlu7
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu4 receptor |
7E9H |
grm7_human |
|
GPR52 |
2022-06-19 |
Inactive |
Yes
|
GPR52
|
GPR52
|
A orphans |
A (Rhodopsin) |
Human |
GPR52 |
6LI1 |
6li1 |
|
ADGRE1 |
2022-06-19 |
Active |
No
|
AGRE1
|
ADGRE1
|
ADGRE |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agre1_human |
|
mGlu5 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM5
|
mGlu5
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
4OO9 |
4oo9 |
|
RXFP1 |
2022-06-19 |
Inactive |
No
|
RXFP1
|
RXFP1
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
A1 receptor |
5UEN |
rxfp1_human |
|
GPR158 |
2022-06-19 |
Active |
No
|
GP158
|
GPR158
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
7C7Q |
gp158_human |
|
TAS2R10 |
2022-06-19 |
Intermediate |
No
|
T2R10
|
TAS2R10
|
Taste 2 |
T (Taste 2) |
Human |
MC4 receptor |
6W25 |
t2r10_human |
|
ADGRE3 |
2022-06-19 |
Intermediate |
No
|
AGRE3
|
ADGRE3
|
ADGRE |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agre3_human |
|
SMO |
2022-06-20 |
Inactive |
Yes
|
SMO
|
SMO
|
Frizzled |
F (Frizzled) |
Human |
SMO |
5V57 |
5v57 |
|
ADGRE4P |
2022-06-19 |
Intermediate |
No
|
AGRE4
|
ADGRE4P
|
ADGRE |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agre4_human |
|
GPR183 |
2022-06-19 |
Inactive |
No
|
GP183
|
GPR183
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
gp183_human |
|
B2 receptor |
2022-06-19 |
Intermediate |
No
|
BKRB2
|
B2
|
Bradykinin |
A (Rhodopsin) |
Human |
GPR183 |
7TUY |
bkrb2_human |
|
ADGRL2 |
2022-06-19 |
Inactive |
No
|
AGRL2
|
ADGRL2
|
ADGRL |
B2 (Adhesion) |
Human |
CRF1 receptor |
4K5Y |
agrl2_human |
|
apelin receptor |
2022-06-19 |
Inactive |
Yes
|
APJ
|
apelin
|
Apelin |
A (Rhodopsin) |
Human |
apelin receptor |
5VBL |
5vbl |
|
A3 receptor |
2022-06-19 |
Inactive |
No
|
AA3R
|
A3
|
Adenosine |
A (Rhodopsin) |
Human |
A1 receptor |
5UEN |
aa3r_human |
|
CXCR3 |
2022-06-19 |
Inactive |
No
|
CXCR3
|
CXCR3
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
cxcr3_human |
|
mGlu5 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM5
|
mGlu5
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu5 receptor |
7FD9 |
7fd9 |
|
M1 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM1
|
M1
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M1 receptor |
6ZG9 |
6zg9 |
|
GPR161 |
2022-06-19 |
Inactive |
No
|
GP161
|
GPR161
|
A orphans |
A (Rhodopsin) |
Human |
α1B-adrenoceptor |
7B6W |
gp161_human |
|
FZD10 |
2022-06-19 |
Active |
No
|
FZD10
|
FZD10
|
Frizzled |
F (Frizzled) |
Human |
FZD7 |
7EVW |
fzd10_human |
|
motilin receptor |
2022-06-19 |
Active |
No
|
MTLR
|
motilin
|
Motilin |
A (Rhodopsin) |
Human |
ghrelin receptor |
7NA7 |
mtlr_human |
|
Rhodopsin |
2022-06-19 |
Inactive |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
3C9M |
3c9m |
|
TAAR2 |
2022-06-19 |
Inactive |
No
|
TAAR2
|
TAAR2
|
A orphans |
A (Rhodopsin) |
Human |
α2A-adrenoceptor |
6KUX |
taar2_human |
|
NK3 receptor |
2022-06-19 |
Active |
No
|
NK3R
|
NK3
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
7P00 |
nk3r_human |
|
AT1 receptor |
2022-06-19 |
Active |
Yes
|
AGTR1
|
AT1
|
Angiotensin |
A (Rhodopsin) |
Human |
AT1 receptor |
6OS2 |
6os2 |
|
A2A receptor |
2022-06-19 |
Active |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
4UHR |
4uhr |
|
GPR12 |
2022-06-19 |
Intermediate |
No
|
GPR12
|
GPR12
|
A orphans |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
gpr12_human |
|
GPR146 |
2022-06-19 |
Inactive |
No
|
GP146
|
GPR146
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
gp146_human |
|
mGlu7 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM7
|
mGlu7
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu7 receptor |
7EPC |
7epc |
|
ADGRA2 |
2022-06-19 |
Intermediate |
No
|
AGRA2
|
ADGRA2
|
ADGRA |
B2 (Adhesion) |
Human |
GLP-1 receptor |
5NX2 |
agra2_human |
|
PAR3 |
2022-06-19 |
Intermediate |
No
|
PAR3
|
PAR3
|
Proteinase-activated |
A (Rhodopsin) |
Human |
PAR2 |
5NDD |
par3_human |
|
succinate receptor |
2022-06-19 |
Inactive |
No
|
SUCR1
|
succinate
|
Succinate |
A (Rhodopsin) |
Human |
apelin receptor |
5VBL |
sucr1_human |
|
5-HT4 receptor |
2022-06-19 |
Intermediate |
No
|
5HT4R
|
5-HT4
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht4r_human |
|
PrRP receptor |
2022-06-19 |
Active |
No
|
PRLHR
|
PrRP
|
Prolactin-releasing peptide |
A (Rhodopsin) |
Human |
OX2 receptor |
7L1V |
prlhr_human |
|
5-HT2A receptor |
2022-06-19 |
Inactive |
Yes
|
5HT2A
|
5-HT2A
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6A93 |
6a93 |
|
CCK1 receptor |
2022-06-19 |
Intermediate |
No
|
CCKAR
|
CCK1
|
Cholecystokinin |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
cckar_human |
|
CaS receptor |
2022-06-19 |
Inactive |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7DTU |
7dtu |
|
GPBA receptor |
2022-06-19 |
Intermediate |
No
|
GPBAR
|
GPBA
|
Bile acid |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
gpbar_human |
|
GPR12 |
2022-06-19 |
Inactive |
No
|
GPR12
|
GPR12
|
A orphans |
A (Rhodopsin) |
Human |
LPA1 receptor |
4Z35 |
gpr12_human |
|
LGR5 |
2022-06-19 |
Active |
No
|
LGR5
|
LGR5
|
A orphans |
A (Rhodopsin) |
Human |
LH receptor |
7FIG |
lgr5_human |
|
ADGRG7 |
2022-06-19 |
Active |
No
|
AGRG7
|
ADGRG7
|
ADGRG |
B2 (Adhesion) |
Human |
ADGRG4 |
7WUJ |
agrg7_human |
|
ETA receptor |
2022-06-19 |
Active |
No
|
EDNRA
|
ETA
|
Endothelin |
A (Rhodopsin) |
Human |
ghrelin receptor |
7NA7 |
ednra_human |
|
5-HT6 receptor |
2022-06-19 |
Intermediate |
No
|
5HT6R
|
5-HT6
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht6r_human |
|
GPR32 |
2022-06-19 |
Inactive |
No
|
GPR32
|
GPR32
|
A orphans |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
gpr32_human |
|
CRF2 receptor |
2022-06-19 |
Inactive |
No
|
CRFR2
|
CRF2
|
Corticotropin-releasing factor |
B1 (Secretin) |
Human |
CRF1 receptor |
4K5Y |
crfr2_human |
|
NPFF2 receptor |
2022-06-19 |
Intermediate |
No
|
NPFF2
|
NPFF2
|
Neuropeptide FF/neuropeptide AF |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
npff2_human |
|
CB1 receptor |
2022-06-19 |
Inactive |
Yes
|
CNR1
|
CB1
|
Cannabinoid |
A (Rhodopsin) |
Human |
CB1 receptor |
5U09 |
5u09 |
|
CaS receptor |
2022-06-19 |
Inactive |
Yes
|
CASR
|
CaS
|
Calcium-sensing |
C (Glutamate) |
Human |
CaS receptor |
7M3J |
7m3j |
|
GPR151 |
2022-06-19 |
Intermediate |
No
|
GP151
|
GPR151
|
A orphans |
A (Rhodopsin) |
Human |
succinate receptor |
6RNK |
gp151_human |
|
P2Y2 receptor |
2022-06-19 |
Active |
No
|
P2RY2
|
P2Y2
|
P2Y |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
p2ry2_human |
|
glucagon receptor |
2022-06-19 |
Intermediate |
No
|
GLR
|
glucagon
|
Glucagon |
B1 (Secretin) |
Human |
GLP-1 receptor |
5NX2 |
glr_human |
|
H3 receptor |
2022-06-19 |
Intermediate |
No
|
HRH3
|
H3
|
Histamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
hrh3_human |
|
NK1 receptor |
2022-06-19 |
Inactive |
Yes
|
NK1R
|
NK1
|
Tachykinin |
A (Rhodopsin) |
Human |
NK1 receptor |
6HLL |
6hll |
|
GPR176 |
2022-06-19 |
Inactive |
No
|
GP176
|
GPR176
|
A orphans |
A (Rhodopsin) |
Human |
OX2 receptor |
5WQC |
gp176_human |
|
GPR174 |
2022-06-19 |
Inactive |
No
|
GP174
|
GPR174
|
A orphans |
A (Rhodopsin) |
Human |
CXCR2 |
6LFL |
gp174_human |
|
ETB receptor |
2022-06-19 |
Active |
No
|
EDNRB
|
ETB
|
Endothelin |
A (Rhodopsin) |
Human |
ghrelin receptor |
7NA7 |
ednrb_human |
|
OX2 receptor |
2022-06-19 |
Inactive |
Yes
|
OX2R
|
OX2
|
Orexin |
A (Rhodopsin) |
Human |
OX2 receptor |
5WQC |
5wqc |
|
GPR153 |
2022-06-19 |
Inactive |
No
|
GP153
|
GPR153
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2A receptor |
6A94 |
gp153_human |
|
β3-adrenoceptor |
2022-06-19 |
Inactive |
No
|
ADRB3
|
β3
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
adrb3_human |
|
GPR139 |
2022-06-19 |
Inactive |
No
|
GP139
|
GPR139
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2C receptor |
6BQH |
gp139_human |
|
CXCR4 |
2022-06-19 |
Inactive |
Yes
|
CXCR4
|
CXCR4
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR4 |
4RWS |
4rws |
|
Rhodopsin |
2022-06-19 |
Active |
Yes
|
OPSD
|
Rhodopsin
|
Opsins |
A (Rhodopsin) |
Bovine |
Rhodopsin |
6FKB |
6fkb |
|
GPR37 |
2022-06-19 |
Intermediate |
No
|
GPR37
|
GPR37
|
A orphans |
A (Rhodopsin) |
Human |
LPA6 receptor |
5XSZ |
gpr37_human |
|
LPA3 receptor |
2022-06-19 |
Intermediate |
No
|
LPAR3
|
LPA3
|
Lysophospholipid (LPA) |
A (Rhodopsin) |
Human |
MC4 receptor |
6W25 |
lpar3_human |
|
GPR22 |
2022-06-19 |
Intermediate |
No
|
GPR22
|
GPR22
|
A orphans |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
gpr22_human |
|
SST3 receptor |
2022-06-19 |
Active |
No
|
SSR3
|
SST3
|
Somatostatin |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
ssr3_human |
|
calcitonin receptor-like receptor |
2022-06-19 |
Inactive |
Yes
|
CALRL
|
calcitonin-like
|
Calcitonin |
B1 (Secretin) |
Human |
calcitonin receptor-like receptor |
7KNT |
7knt |
|
5-HT1E receptor |
2022-06-19 |
Intermediate |
No
|
5HT1E
|
5-HT1E
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
5ht1e_human |
|
A2A receptor |
2022-06-19 |
Inactive |
Yes
|
AA2AR
|
A2A
|
Adenosine |
A (Rhodopsin) |
Human |
A2A receptor |
6WQA |
6wqa |
|
EP3 receptor |
2022-06-19 |
Active |
Yes
|
PE2R3
|
EP3
|
Prostanoid |
A (Rhodopsin) |
Human |
EP3 receptor |
6AK3 |
6ak3 |
|
GPR31 |
2022-06-19 |
Active |
No
|
GPR31
|
GPR31
|
A orphans |
A (Rhodopsin) |
Human |
SST2 receptor |
7T10 |
gpr31_human |
|
MC4 receptor |
2022-06-19 |
Inactive |
No
|
MC4R
|
MC4
|
Melanocortin |
A (Rhodopsin) |
Human |
S1P1 receptor |
3V2Y |
mc4r_human |
|
GPRC5A |
2022-06-19 |
Intermediate |
No
|
RAI3
|
GPRC5A
|
C Orphans |
C (Glutamate) |
Human |
mGlu5 receptor |
6N51 |
rai3_human |
|
GAL3 receptor |
2022-06-19 |
Inactive |
No
|
GALR3
|
GAL3
|
Galanin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
galr3_human |
|
A1 receptor |
2022-06-19 |
Inactive |
Yes
|
AA1R
|
A1
|
Adenosine |
A (Rhodopsin) |
Human |
A1 receptor |
5UEN |
5uen |
|
ADGRL1 |
2022-06-19 |
Active |
No
|
AGRL1
|
ADGRL1
|
ADGRL |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agrl1_human |
|
NOP receptor |
2022-06-19 |
Inactive |
Yes
|
OPRX
|
NOP
|
Opioid |
A (Rhodopsin) |
Human |
NOP receptor |
4EA3 |
4ea3 |
|
EP2 receptor |
2022-06-19 |
Inactive |
No
|
PE2R2
|
EP2
|
Prostanoid |
A (Rhodopsin) |
Human |
EP4 receptor |
5YWY |
pe2r2_human |
|
RXFP3 |
2022-06-19 |
Inactive |
No
|
RL3R1
|
RXFP3
|
Relaxin family peptide |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
rl3r1_human |
|
mGlu3 receptor |
2022-06-19 |
Inactive |
Yes
|
GRM3
|
mGlu3
|
Metabotropic glutamate |
C (Glutamate) |
Human |
mGlu3 receptor |
7WI8 |
7wi8 |
|
SST3 receptor |
2022-06-19 |
Inactive |
No
|
SSR3
|
SST3
|
Somatostatin |
A (Rhodopsin) |
Human |
κ receptor |
4DJH |
ssr3_human |
|
TAS2R19 |
2022-06-19 |
Intermediate |
No
|
T2R19
|
TAS2R19
|
Taste 2 |
T (Taste 2) |
Human |
CysLT1 receptor |
6RZ4 |
t2r19_human |
|
GPR156 |
2022-06-19 |
Active |
No
|
GP156
|
GPR156
|
C Orphans |
C (Glutamate) |
Human |
GABAB2 |
7C7Q |
gp156_human |
|
5-HT6 receptor |
2022-06-19 |
Inactive |
No
|
5HT6R
|
5-HT6
|
5-Hydroxytryptamine |
A (Rhodopsin) |
Human |
β1-adrenoceptor |
7BVQ |
5ht6r_human |
|
MAS1 |
2022-06-19 |
Inactive |
No
|
MAS
|
MAS1
|
A orphans |
A (Rhodopsin) |
Human |
AT1 receptor |
4ZUD |
mas_human |
|
β1-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB1
|
β1
|
Adrenoceptors |
A (Rhodopsin) |
Wild turkey |
β1-adrenoceptor |
2YCZ |
2ycz |
|
CCR8 |
2022-06-19 |
Active |
No
|
CCR8
|
CCR8
|
Chemokine |
A (Rhodopsin) |
Human |
CCR1 |
7VL9 |
ccr8_human |
|
succinate receptor |
2022-06-19 |
Intermediate |
Yes
|
SUCR1
|
succinate
|
Succinate |
A (Rhodopsin) |
Rat |
succinate receptor |
6Z10 |
6z10 |
|
β2-adrenoceptor |
2022-06-19 |
Inactive |
Yes
|
ADRB2
|
β2
|
Adrenoceptors |
A (Rhodopsin) |
Human |
β2-adrenoceptor |
4GBR |
4gbr |
|
ADGRL2 |
2022-06-19 |
Active |
No
|
AGRL2
|
ADGRL2
|
ADGRL |
B2 (Adhesion) |
Human |
ADGRL3 |
7SF7 |
agrl2_human |
|
glucagon receptor |
2022-06-19 |
Inactive |
Yes
|
GLR
|
glucagon
|
Glucagon |
B1 (Secretin) |
Human |
glucagon receptor |
5YQZ |
5yqz |
|
CXCR4 |
2022-06-19 |
Inactive |
Yes
|
CXCR4
|
CXCR4
|
Chemokine |
A (Rhodopsin) |
Human |
CXCR4 |
3OE0 |
3oe0 |
|
TAS2R9 |
2022-06-19 |
Active |
No
|
TA2R9
|
TAS2R9
|
Taste 2 |
T (Taste 2) |
Human |
H1 receptor |
7DFL |
ta2r9_human |
|
D1 receptor |
2022-06-19 |
Intermediate |
No
|
DRD1
|
D1
|
Dopamine |
A (Rhodopsin) |
Human |
5-HT2B receptor |
5TVN |
drd1_human |
|
M1 receptor |
2022-06-19 |
Inactive |
Yes
|
ACM1
|
M1
|
Acetylcholine (muscarinic) |
A (Rhodopsin) |
Human |
M1 receptor |
6ZFZ |
6zfz |
|
secretin receptor |
2022-06-19 |
Inactive |
No
|
SCTR
|
secretin
|
Glucagon |
B1 (Secretin) |
Human |
PTH1 receptor |
6FJ3 |
sctr_human |
|
glucagon receptor |
2022-06-19 |
Inactive |
Yes
|
GLR
|
glucagon
|
Glucagon |
B1 (Secretin) |
Human |
glucagon receptor |
4L6R |
4l6r |
|
ACKR4 |
2022-06-19 |
Active |
No
|
ACKR4
|
ACKR4
|
Chemokine |
A (Rhodopsin) |
Human |
CCR6 |
6WWZ |
ackr4_human |
|
ADGRL2 |
2022-06-19 |
Intermediate |
No
|
AGRL2
|