Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
oprm_mouse 3.32x32 147 TM3 D => A N/A N/A Befort K et al (1996)
oprm_mouse 2.50x50 114 TM2 D => A N/A N/A Chakrabarti S et al (1997)
oprm_mouse 2.50x50 114 TM2 D => N N/A N/A Pil J et al (2003)
oprm_mouse 2.50x50 114 TM2 D => N N/A N/A Bot G et al (1998)
oprm_mouse 4.54x54 196 TM4 S => A N/A N/A Claude-Geppert PA et al (2005)
oprm_mouse 4.54x54 196 TM4 S => L N/A N/A Claude-Geppert PA et al (2005)
oprm_mouse 7.35x34 318 TM7 W => Y N/A N/A Ulens C et al (2001)
oprm_mouse 7.36x35 319 TM7 H => Y N/A N/A Ulens C et al (2001)
oprm_mouse 7.43x42 326 TM7 Y => F N/A N/A Pil J et al (2003)
oprm_mouse 7.44x43 327 TM7 T => A N/A N/A Claude-Geppert PA et al (2005)
oprm_mouse 7.46x46 329 TM7 S => A N/A N/A Pil J et al (2003)
oprm_mouse 7.47x47 330 TM7 C => A N/A N/A Claude-Geppert PA et al (2005)
oprm_mouse 7.47x47 330 TM7 C => S N/A N/A Claude-Geppert PA et al (2005)
oprm_mouse 7.49x49 332 TM7 N => D N/A N/A Pil J et al (2003)
oprm_mouse 8.58x58 351 H8 C => L N/A N/A Zhang L et al (2006)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 T T K Y R Q G S I D C T L T F S H ECL2ICL3 R M L S G ICL3ECL3 T I P E ECL3N-term M D S S A G P G N I S D C S D P L A P A S C S P A P G S W L N L S H V D G N Q S D P C G P N R T G L G G S H S L C P Q T G S P S N-termC-term P T S S T I E Q Q N S A R I R Q N T R E H P S T A N T V D R T N H Q L E N L E A E T A P L P C-term M V T A I T I M A L Y S I V C V V G L F G N F L V M Y V I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S V N Y L M G G N I L C K I V I S I D Y Y N M F T S I F T L C T M S V D R Y I A V C H T P R N A K I V N V C N W I L S S A I G L P V M F M A P T W Y W E N L L K I C V F I F A F I M P V L I I T V C Y G L M I L R L K S V S K E K D R N L R R I T R M V L V V V A V F I V C W T P I H I Y V I I K A L I T T F Q T V S W H F C I A L G Y T N S C L N P V L Y A F L D E N F R E F K R C F C I
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
F N G F L G V V C V I S Y L A M I T I A 1 F N L A L A D A L A T S T L P F Q S V N 2 T C L T F I S T F M N Y Y D I S I V I K 3 A K I V N V C N W I L S S A I G L P V M 4 Y C V T I I L V P M I F A F I F V C I K L 5 L V V V A V F I V C W T P I H I Y V I I 6 V P N L C S N T Y G L A I C F H W S V 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
μ receptor
TM2
2x50 2.50x50 D114
TM3
3x32 3.32x32 D147
TM4
4x54 4.54x54 S196
TM7
7x34 7.35x34 W318
7x35 7.36x35 H319
7x42 7.43x42 Y326
7x43 7.44x43 T327
7x46 7.46x46 S329
7x47 7.47x47 C330
7x49 7.49x49 N332
H8
8x58 8.58x58 C351